SCHEMBL10399407

SCHEMBL10399407

Nc1cc(Nc2ccccc2)nc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.72
THPO P40225 2/20 0.72
CYP2C19 P33261 2/20 0.72
ADORA2A P29274 2/20 0.72
ADORA2B P29275 1/20 0.72
MEN1 O00255 1/20 0.72
CYP2D6 P10635 1/20 0.72
CYP2C9 P11712 1/20 0.72
KMT2A Q03164 1/20 0.72
BLM P54132 1/20 0.72
LMNA P02545 2/20 0.64
ALDH1A1 P00352 1/20 0.64
GLA P06280 1/20 0.64
PMP22 Q01453 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
NPC1 O15118 1/20 0.64
NPY1R P25929 1/20 0.64
HTT P42858 1/20 0.64
NPY2R P49146 1/20 0.64
RAB9A P51151 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10399798 0.85 PGK1 (0.70) THPOADORA2AADORA2BSLC29A1TSHR
SCHEMBL10399490 0.84 PI4KA (0.57) CYP1A2THPOCYP2C19ADORA2AADORA2B
SCHEMBL29387702 0.84 CYP1A2 (1.00) CYP1A2THPOCYP2C19ADORA2AADORA2B
SCHEMBL725689 0.84 CYP1A2 (1.00) CYP1A2THPOCYP2C19ADORA2AADORA2B
SCHEMBL725690 0.84 CYP1A2 (1.00) CYP1A2THPOCYP2C19ADORA2AADORA2B
SCHEMBL4808305 0.84 CYP1A2 (0.73) CYP1A2THPOCYP2C19ADORA2AADORA2B
SCHEMBL29753859 0.84 CYP1A2 (1.00) CYP1A2THPOCYP2C19ADORA2AADORA2B
SCHEMBL10399357 0.83 ADORA2A (0.68) ADORA2AADORA2BSLC29A1ADORA3ADORA1
SCHEMBL10399488 0.82 ADORA3 (0.62) ADORA2AADORA2BADORA3ADORA1
SCHEMBL10625871 0.81 ADORA2A (0.70) CYP1A2THPOCYP2C19ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4977144-A ADENOSINE AGONISTS CIBA-GEIGY CORPORATION (US) 1990-12-11 US disclosed
EP-0354180-A2 Certain imidazo[4,5-b]pyridine derivatives CIBA-GEIGY AG (CH) 1990-02-07 EP disclosed