SCHEMBL10399798

SCHEMBL10399798

Nc1cc(NCCc2ccccc2)nc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.74

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PGK1 P00558 3/20 0.70
PGK2 P07205 3/20 0.70
ADORA3 P0DMS8 5/20 0.67
ADORA1 P30542 3/20 0.67
ADORA2A P29274 3/20 0.67
NFKB1 P19838 1/20 0.67
THPO P40225 1/20 0.67
TSHR P16473 1/20 0.67
ADORA2B P29275 2/20 0.62
SLC29A1 Q99808 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10399357 0.95 ADORA2A (0.68) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL10399504 0.91 ADORA2A (0.64) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL10399499 0.91 ADORA2A (0.63) PGK1PGK2ADORA2ATSHRADORA2B
SCHEMBL10399501 0.90 ADORA2A (0.76) PGK1PGK2ADORA3ADORA1ADORA2A
Hydrochloric Acid SCHEMBL10399464 0.90 ADORA2A (0.63) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL10398375 0.89 ADORA2A (0.66) ADORA2ATSHRADORA2B
SCHEMBL10398379 0.88 SLC29A1 (0.60) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL8373469 0.85 ADORA2A (0.82) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL10587027 0.85 ADORA2A (0.82) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL10399407 0.85 CYP1A2 (0.72) ADORA3ADORA1ADORA2ANFKB1THPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4977144-A ADENOSINE AGONISTS CIBA-GEIGY CORPORATION (US) 1990-12-11 US claimed
EP-0354180-A2 Certain imidazo[4,5-b]pyridine derivatives CIBA-GEIGY AG (CH) 1990-02-07 EP claimed
US-4977144-A ADENOSINE AGONISTS CIBA-GEIGY CORPORATION (US) 1990-12-11 US disclosed