SCHEMBL10399592

SCHEMBL10399592

CN(C)/C=C1\C(=O)Nc2cccc(Cl)c21

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 14/20 0.62
SMN1; SMN2 Q16637 1/20 0.59
CES1 P23141 1/20 0.56
ALDH1A1 P00352 2/20 0.45
MAPT P10636 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10399594 1.00 TGM2 (0.62) TGM2SMN1; SMN2CES1ALDH1A1MAPT
SCHEMBL13244119 0.83 SMN1; SMN2 (0.61) TGM2SMN1; SMN2ALDH1A1MAPTNPSR1
SCHEMBL2512919 0.81 SMN1; SMN2 (0.59) TGM2SMN1; SMN2CES1ALDH1A1MAPT
SCHEMBL12200893 0.81 SMN1; SMN2 (0.59) TGM2SMN1; SMN2CES1ALDH1A1MAPT
SCHEMBL10399806 0.76 TGM2 (0.64) TGM2SMN1; SMN2CES1ALDH1A1MAPT
SCHEMBL10399808 0.76 TGM2 (0.64) TGM2SMN1; SMN2CES1ALDH1A1MAPT
SCHEMBL397664 0.75 SMN1; SMN2 (1.00) TGM2SMN1; SMN2ALDH1A1MAPTNPSR1
SCHEMBL11892099 0.75 SMN1; SMN2 (1.00) TGM2SMN1; SMN2ALDH1A1MAPTNPSR1
SCHEMBL397665 0.75 SMN1; SMN2 (1.00) TGM2SMN1; SMN2ALDH1A1MAPTNPSR1
SCHEMBL30716604 0.72 CES1 (1.00) TGM2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4977178-A Method of treating anxiety and depression with 1-phenyl-2(1H,3H)-indolone psycho-therapeutic agents PFIZER INC. (US) 1990-12-11 US disclosed
US-4879391-A 1-Phenyl-2(1H,3H)-indolone psychotherapeutic agents PFIZER INC. (US) 1989-11-07 US disclosed
US-4861880-A 1-phenyl-2(1H,3H)-indolone psycho-therapeutic agents PFIZER INC. (US) 1989-08-29 US disclosed
US-4476307-A Heteroylidene indolone compounds PFIZER INC. (US) 1984-10-09 US disclosed
EP-0104860-A1 1-Phenyl-2(1H,3H)-indolone psycho-therapeutic agents PFIZER INC. (US) 1984-04-04 EP disclosed