SCHEMBL10399501

SCHEMBL10399501

Nc1cc(NCCc2ccc(CCC(=O)O)cc2)nc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.76

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.76
ADORA2B P29275 3/20 0.76
ADORA3 P0DMS8 2/20 0.58
ADORA1 P30542 2/20 0.58
PGK1 P00558 3/20 0.58
PGK2 P07205 3/20 0.58
LMNA P02545 1/20 0.58
MAPT P10636 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
CYP3A4 P08684 1/20 0.58
TSHR P16473 1/20 0.58
MAPK1 P28482 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10399798 0.90 PGK1 (0.70) ADORA2AADORA2BADORA3ADORA1PGK1
SCHEMBL10399504 0.89 ADORA2A (0.64) ADORA2AADORA2BADORA3ADORA1PGK1
SCHEMBL10399499 0.89 ADORA2A (0.63) ADORA2AADORA2BPGK1PGK2LMNA
Hydrochloric Acid SCHEMBL10399464 0.88 ADORA2A (0.63) ADORA2AADORA2BADORA3ADORA1PGK1
SCHEMBL10399463 0.86 ADORA2A (0.58) ADORA2AADORA2BADORA3ADORA1LMNA
SCHEMBL9762945 0.86 ADORA2A (1.00) ADORA2AADORA2BADORA3ADORA1TSHR
SCHEMBL10588368 0.86 ADORA2A (1.00) ADORA2AADORA2BADORA3ADORA1TSHR
SCHEMBL10398375 0.86 ADORA2A (0.66) ADORA2AADORA2BLMNAMAPTNPSR1
Hydrochloric Acid SCHEMBL9762842 0.86 ADORA2A (0.98) ADORA2AADORA2BADORA3ADORA1TSHR
SCHEMBL10399357 0.85 ADORA2A (0.68) ADORA2AADORA2BADORA3ADORA1PGK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4977144-A ADENOSINE AGONISTS CIBA-GEIGY CORPORATION (US) 1990-12-11 US disclosed
EP-0354180-A2 Certain imidazo[4,5-b]pyridine derivatives CIBA-GEIGY AG (CH) 1990-02-07 EP disclosed