SCHEMBL10400985

SCHEMBL10400985

CCOC(=O)Nc1nc(C)ncc1C(=O)OCC

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FOS P01100 7/20 0.60
JUN P05412 7/20 0.60
NFKB1 P19838 7/20 0.60
NFKB2 Q00653 7/20 0.60
RELA Q04206 7/20 0.60
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 2/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
AGTR1 P30556 1/20 0.45
AGTR2 P50052 1/20 0.45
CSNK1D P48730 1/20 0.45
ALOX15 P16050 1/20 0.45
HSP90AA1 P07900 1/20 0.45
SYK P43405 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15624862 0.85 ALDH1A1 (0.60) FOSJUNNFKB1NFKB2RELA
SCHEMBL19320623 0.84 FOS (0.58) FOSJUNNFKB1NFKB2RELA
SCHEMBL9496451 0.80 ALDH1A1 (0.51) FOSJUNNFKB1NFKB2RELA
SCHEMBL17466945 0.78 FOS (0.53) FOSJUNNFKB1NFKB2RELA
SCHEMBL1627061 0.78 FOS (0.53) FOSJUNNFKB1NFKB2RELA
SCHEMBL1669574 0.78 RAB9A (0.56) FOSJUNNFKB1NFKB2RELA
SCHEMBL30996914 0.78 RAB9A (0.56) FOSJUNNFKB1NFKB2RELA
SCHEMBL959574 0.76 CSNK1D (0.54) FOSJUNNFKB1NFKB2RELA
SCHEMBL3283452 0.75 ALDH1A1 (0.50) FOSJUNNFKB1NFKB2RELA
SCHEMBL6604256 0.75 SMN1; SMN2 (0.63) NFKB1NFKB2RELAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4950648-A SUBSTITUTED PYRIDO(2,3-D) OR PYRIMIDO(4,5-D) PYRIMIDINE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1990-08-21 US disclosed
EP-0316668-A2 Use of a tetrahydro-pyrido(2,3-d)pyrimidine for obtaining an analgetic agent MERCK PATENT GmbH (DE) 1989-05-24 EP disclosed