SCHEMBL10401634

SCHEMBL10401634

N#Cc1cc(Cl)c(Cl)cc1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.44
TSHR P16473 3/20 0.42
POLB P06746 1/20 0.42
ALDH1A1 P00352 3/20 0.41
CASP1 P29466 2/20 0.41
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 2/20 0.40
HSD17B10 Q99714 2/20 0.40
AKR1C4 P17516 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
HTT P42858 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
EIF4E P06730 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23699498 0.85 MRGPRX4 (0.41) MRGPRX4TSHRPOLBALDH1A1CASP1
SCHEMBL16968396 0.84 KDM4E (0.50) MRGPRX4ALDH1A1SMN1; SMN2KDM4EHSD17B10
SCHEMBL8576784 0.81 CA12 (0.46) MRGPRX4TSHRALDH1A1KDM4EHSD17B10
SCHEMBL11116363 0.80 KDM4E (0.47) MRGPRX4ALDH1A1SMN1; SMN2KDM4EHSD17B10
SCHEMBL8572624 0.79 CISD1 (0.66) ALDH1A1
SCHEMBL31171383 0.78 CA12 (0.46) MRGPRX4TSHRPOLBALDH1A1CASP1
SCHEMBL11255716 0.77 GAA (0.49) ALDH1A1SMN1; SMN2KDM4EHSD17B10HTT
SCHEMBL8304252 0.77 KEAP1 (0.44) MRGPRX4TSHRPOLBALDH1A1CASP1
SCHEMBL8299931 0.77 ALDH1A1 (0.42) MRGPRX4TSHRALDH1A1CASP1TP53
SCHEMBL23699456 0.77 TRPV4 (0.43) MRGPRX4TSHRPOLBALDH1A1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4946858-A ANTIDIABETIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1990-08-07 US disclosed
US-4900739-A ANTIDIABETIC AGENTS AMERICAN HOME PRODUCTS CORP. (US) 1990-02-13 US disclosed
US-4317929-A Tetraphenylketazines and isoindolinone pigments obtained therefrom CIBA-GEIGY CORPORATION (US) 1982-03-02 US disclosed
US-4231931-A YELLOW TO RED HUES CIBA-GEIGY CORPORATION (US) 1980-11-04 US disclosed