SCHEMBL10405409

SCHEMBL10405409

Nc1nc(O)c2cc(CCCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)ccc2n1

nearest known ligand 0.63

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHFR P00374 9/20 0.63
GART P22102 6/20 0.59
FOLR2 P14207 2/20 0.59
FOLR1 P15328 2/20 0.59
SLC46A1 Q96NT5 2/20 0.59
SLC19A1 P41440 1/20 0.59
ATIC P31939 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9446115 0.91 DHFR (0.75) DHFRGARTFOLR2FOLR1SLC46A1
SCHEMBL9263780 0.87 GART (0.67) DHFRGARTFOLR2FOLR1SLC46A1
SCHEMBL24629143 0.87 DHFR (0.55) DHFRGART
SCHEMBL25904683 0.86 DHFR (0.54) DHFRGART
SCHEMBL12717668 0.86 DHFR (0.72) DHFR
SCHEMBL12717676 0.86 DHFR (0.72) DHFR
SCHEMBL9339136 0.85 GART (0.68) DHFRGARTFOLR2FOLR1SLC46A1
SCHEMBL9844787 0.84 DHFR (0.61) DHFRGARTFOLR2FOLR1SLC46A1
SCHEMBL6337570 0.84 DHFR (0.77) DHFRGARTFOLR2FOLR1SLC46A1
SCHEMBL9844791 0.84 GART (0.73) DHFRGARTFOLR2FOLR1SLC46A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4946846-A ANTITUMOR AGENTS; NONTOXIC TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-08-07 US claimed
US-4946846-A ANTITUMOR AGENTS; NONTOXIC TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-08-07 US disclosed