SCHEMBL1040563

SCHEMBL1040563

O=C(NCc1ccc([N+](=O)[O-])cc1)c1ccc2c(c1)OCO2

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.73
MAPT P10636 5/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
GAA P10253 1/20 0.67
MEN1 O00255 3/20 0.65
KMT2A Q03164 3/20 0.65
LMNA P02545 2/20 0.62
MAPK1 P28482 2/20 0.62
MMP13 P45452 1/20 0.62
POLB P06746 1/20 0.61
P2RX5 Q93086 1/20 0.60
P2RX4 Q99571 1/20 0.60
P2RX7 Q99572 1/20 0.60
P2RX2 Q9UBL9 1/20 0.60
HPGD P15428 1/20 0.60
NPC1 O15118 1/20 0.60
ROCK2 O75116 1/20 0.59
HSP90AA1 P07900 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
HTT P42858 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12443107 0.85 ALDH1A1 (0.81) ALDH1A1MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL108263 0.84 ALDH1A1 (0.92) ALDH1A1MEN1KMT2ALMNAMAPK1
SCHEMBL1042605 0.82 ALDH1A1 (0.74) ALDH1A1SMN1; SMN2MEN1KMT2ALMNA
SCHEMBL647939 0.82 RAB9A (0.84) ALDH1A1MAPTSMN1; SMN2GAAMEN1
SCHEMBL1040562 0.79 MAPT (0.76) ALDH1A1MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL1041554 0.79 ALDH1A1 (0.69) ALDH1A1MEN1KMT2ALMNAMAPK1
SCHEMBL14900330 0.79 ALDH1A1 (0.69) ALDH1A1MAPTGAAMEN1KMT2A
SCHEMBL1042327 0.79 RAB9A (0.78) ALDH1A1MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL15306501 0.79 KMT2A (1.00) ALDH1A1MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL6940835 0.78 ALDH1A1 (0.69) ALDH1A1MAPTSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1480941-B1 UREA DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS AMBRILIA BIOPHARMA INC (CA) 2011-01-26 EP disclosed
EP-1480941-A2 UREA DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS Procyon Biopharma Inc. (CA) 2004-12-01 EP disclosed
WO-2003074467-A2 UREA DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS PROCYON BIOPHARMA INC. (CA) 2003-09-12 WO disclosed
US-6528532-B1 Benzenesulfonamide group PHARMACOR INC. (CA) 2003-03-04 US disclosed