SCHEMBL10405652

SCHEMBL10405652

O=C(O)CCC(=O)c1ccc2c(c1)CCC2.O=S1(=O)Cc2ccc(cc2)N1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 2/20 0.44
WNT3A P56704 2/20 0.44
ALDH1A1 P00352 4/20 0.43
PKM P14618 1/20 0.37
TSHR P16473 1/20 0.37
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
MAPT P10636 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
PARP1 P09874 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR7 P34969 1/20 0.35
DRD3 P35462 1/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10405645 0.87 CTNNB1 (0.41) CTNNB1WNT3AALDH1A1MAPTTDP1
SCHEMBL10406948 0.86 ALDH1A1 (0.41) CTNNB1WNT3AALDH1A1MAPTTDP1
SCHEMBL6504541 0.81 ALDH1A1 (0.62) CTNNB1WNT3AALDH1A1PKMTSHR
SCHEMBL10406411 0.81 FFAR4 (0.42) ALDH1A1TSHRRXRARXRBRXRG
SCHEMBL10405668 0.81 CTNNB1 (0.49) CTNNB1WNT3AALDH1A1PPARGPPARA
SCHEMBL10405650 0.81 ALDH1A1 (0.39) ALDH1A1MAPTRXRARXRBRXRG
SCHEMBL10406926 0.80 RXRB (0.46) ALDH1A1TSHRMAPTRXRARXRB
SCHEMBL10405870 0.80 RXRA (0.34) ALDH1A1TSHRRXRARXRBRXRG
SCHEMBL817710 0.78 CTNNB1 (0.66) CTNNB1WNT3AALDH1A1PKMTSHR
SCHEMBL10406130 0.78 RAB9A (0.37) CTNNB1WNT3AALDH1A1MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4929754-A CARDIOVASCULAR DISORDERS, ANTICOAGULANTS, ANTITUMOR AGENTS DR. KARL THOMAE GMBH (DE) 1990-05-29 US claimed
US-4929754-A CARDIOVASCULAR DISORDERS, ANTICOAGULANTS, ANTITUMOR AGENTS DR. KARL THOMAE GMBH (DE) 1990-05-29 US disclosed
US-4820705-A ANTITUMOR, CARDIOVASCULR DISORDERS DR. KARL THOMAE GMBH (DE) 1989-04-11 US disclosed