SCHEMBL10409092

SCHEMBL10409092

CN(C)CCc1ccc(O)c2nc(C(F)(F)F)[nH]c12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.41
HTR2A P28223 5/20 0.38
CSNK2A1 P68400 2/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
HTR2C P28335 4/20 0.35
HTR2B P41595 2/20 0.35
HTR7 P34969 2/20 0.35
DRD1 P21728 1/20 0.35
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35
HTR1E P28566 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
DRD3 P35462 1/20 0.35
HTR5A P47898 1/20 0.35
HTR6 P50406 1/20 0.35
MAPT P10636 1/20 0.34
NEK1 Q96PY6 1/20 0.34
TAAR1 Q96RJ0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688999 0.90 HTR1A (0.41) HTR1AHTR2ACSNK2A1CSNK2A2CSNK2B
SCHEMBL10409117 0.82 PDE4B (0.42) HTR1AHTR2ACSNK2A1HTR6
SCHEMBL9688945 0.81 ADRB2 (0.47) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9688843 0.80 HTR1A (0.41) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9688854 0.77 PDE4B (0.47) HTR1AHTR2ACSNK2A1HTR6
SCHEMBL9687970 0.75 HTR1A (0.38) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL10639573 0.74 MAPT (0.44) CSNK2A1CSNK2A2CSNK2BMAPTKDM4E
Hydrochloric Acid SCHEMBL10633457 0.72 MAPT (0.42) CSNK2A1CSNK2A2CSNK2BMAPTKDM4E
SCHEMBL9689133 0.71 HTR1A (0.46) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9688933 0.70 ADRB2 (0.47) HTR1AHTR2AHTR2CHTR2BHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed