SCHEMBL9689133

SCHEMBL9689133

CN(C)CCc1ccc(O)c2nc[nH]c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.46
ALDH1A1 P00352 1/20 0.44
PKM P14618 1/20 0.44
HTR2A P28223 7/20 0.41
HTR2C P28335 6/20 0.41
HTR2B P41595 5/20 0.41
HTR7 P34969 3/20 0.41
HTR6 P50406 3/20 0.41
HTR1B P28222 2/20 0.41
HTR5A P47898 2/20 0.41
DRD1 P21728 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1E P28566 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
DRD3 P35462 1/20 0.41
SLC6A4 P31645 1/20 0.38
MAOA P21397 3/20 0.38
MAOB P27338 2/20 0.38
ADRA2A P08913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689122 0.88 HTR1A (0.46) HTR1AALDH1A1PKMHTR2AHTR2C
SCHEMBL9687926 0.84 HTR1A (0.48) HTR1AALDH1A1PKMHTR2ADRD1
SCHEMBL9689140 0.79 HTR6 (0.47) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9688945 0.75 ADRB2 (0.47) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9689134 0.74 HTR6 (0.50) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9688843 0.74 HTR1A (0.41) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9687915 0.72 HTR1A (0.48) HTR1AALDH1A1PKMHTR2ADRD1
SCHEMBL2267949 0.72 CSNK2A1 (0.41) ALDH1A1PKM
SCHEMBL10409092 0.71 HTR1A (0.41) HTR1AHTR2AHTR2CHTR2BHTR7
Bromide SCHEMBL11357233 0.70 CSNK2A1 (0.40) ALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0189473-B1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1992-05-27 EP disclosed
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed