SCHEMBL10409372

SCHEMBL10409372

CC(C)NCCSc1cccc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 3/20 0.51
NR2E1 Q9Y466 5/20 0.50
IFNAR1 P17181 1/20 0.42
SIGMAR1 Q99720 6/20 0.40
ALDH1A1 P00352 5/20 0.40
ADRB2 P07550 5/20 0.40
ADRB1 P08588 5/20 0.40
LMNA P02545 4/20 0.40
ADRB3 P13945 4/20 0.40
CYP1A2 P05177 3/20 0.40
CYP2D6 P10635 3/20 0.40
SLC6A4 P31645 3/20 0.40
HTR2B P41595 3/20 0.40
HTR2A P28223 3/20 0.40
HTR2C P28335 3/20 0.40
HTR6 P50406 3/20 0.40
MAPK1 P28482 3/20 0.40
SCN1A P35498 2/20 0.40
SLC10A1 Q14973 2/20 0.40
SCN2A Q99250 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10411043 0.98 HTR1B (0.50) HTR1BNR2E1IFNAR1SIGMAR1ALDH1A1
Hydrochloric Acid SCHEMBL11283634 0.76 HTR1B (0.50) HTR1BIFNAR1ALDH1A1LMNAMAPK1
SCHEMBL13601938 0.76 HTR1A (0.43) HTR1BNR2E1HTR1AADRA1ACACNA2D1
SCHEMBL2607777 0.75 IFNAR1 (0.45) IFNAR1ALDH1A1LMNACYP1A2MAPK1
SCHEMBL6293960 0.75 IFNAR1 (0.43) IFNAR1ALDH1A1LMNACYP1A2MAPK1
SCHEMBL2117027 0.74 IFNAR1 (0.44) IFNAR1ALDH1A1LMNACYP1A2MAPK1
SCHEMBL2607673 0.73 TLR8 (0.50) HTR1BIFNAR1ALDH1A1LMNAMAPK1
SCHEMBL10409466 0.72 CNR2 (0.50) HTR1BNR2E1CYP1A2CYP2D6TSHR
SCHEMBL10409411 0.72 BCL2L1 (0.35) SIGMAR1ALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL1493101 0.72 ALDH1A1 (0.44) IFNAR1ALDH1A1LMNACYP1A2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4895840-A ANTIARRHYTHMIA AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1990-01-23 US disclosed
EP-0295010-A1 Derivatives of alkylaminoalkyl ureas and cyanoguanidines A.H. ROBINS COMPANY, INCORPORATED (US) 1988-12-14 EP disclosed
US-4724235-A N-(arylthioalkyl)-N'-(aminoalkyl)ureas useful in the treatment of arrhythmia A. H. ROBINS COMPANY, INCORPORATED (US) 1988-02-09 US disclosed
US-4597902-A TREATMENT OF CARDIAC ARRHYTHMIAS A. H. ROBINS COMPANY, INCORPORATED (US) 1986-07-01 US disclosed
EP-0066415-B1 N-(ARYLTHIOALKYL)-N'-(AMINOALKYL)UREAS A.H. ROBINS COMPANY, INCORPORATED (US) 1985-10-02 EP disclosed
EP-0066415-A2 N-(arylthioalkyl)-N'-(aminoalkyl)ureas A.H. ROBINS COMPANY, INCORPORATED (US) 1982-12-08 EP disclosed