SCHEMBL1041032

SCHEMBL1041032

COCCCN1CCOc2ccc(CO[C@H]3CN(S(=O)(=O)c4ccc(C)cc4)[C@@](CO[SiH3])(C(C)C)C(C(C)C)(C(C)C)[C@H]3c3ccc(CO)cc3)cc21

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.33
CYP2C9 P11712 1/20 0.33
RORC P51449 7/20 0.32
REN P00797 1/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4583099 0.80 CYP2C9 (0.33) KMT2ACYP2C9RORCRENPOLB
SCHEMBL2683799 0.77 KMT2A (0.35) KMT2ACYP2C9RORCRENMEN1
SCHEMBL2683870 0.77 KMT2A (0.35) KMT2ACYP2C9RORCRENMEN1
SCHEMBL5505093 0.75 CYP2C9 (0.33) KMT2ACYP2C9RORCRENMEN1
SCHEMBL1041031 0.75 CYP2C9 (0.33) KMT2ACYP2C9RORCRENMEN1
SCHEMBL2683168 0.74 KMT2A (0.38) KMT2ACYP2C9RORCRENMEN1
SCHEMBL2683813 0.73 KMT2A (0.36) KMT2ACYP2C9RORCRENMEN1
SCHEMBL1036350 0.73 KMT2A (0.37) KMT2ACYP2C9RORCRENMEN1
SCHEMBL3907620 0.73 PKM (0.39) KMT2ACYP2C9RENPOLB
SCHEMBL2682464 0.73 KMT2A (0.36) KMT2ACYP2C9RORCRENMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049514-B1 NITRATE ESTERS OF PIPERIDINES NOVARTIS AG (CH) 2011-01-26 EP disclosed