SCHEMBL10412907

SCHEMBL10412907

Fc1ccc2ccn(Cc3ccccc3)c2c1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.58
APP P05067 4/20 0.53
SNCA P37840 3/20 0.53
HTR2C P28335 2/20 0.53
HTR2A P28223 1/20 0.53
BRD4 O60885 2/20 0.50
P2RX7 Q99572 1/20 0.48
BACE1 P56817 1/20 0.48
CD74 P04233 1/20 0.46
MIF P14174 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.45
HTR7 P34969 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6086002 0.90 HTR2C (0.55) HTR6APPSNCAHTR2CHTR2A
SCHEMBL9584191 0.87 APP (0.53) HTR6APPSNCAHTR2CHTR2A
Quinoline SCHEMBL28080464 0.85 HTR6 (0.52) HTR6APPSNCAHTR2CHTR2A
SCHEMBL6087849 0.85 MAPT (0.53) HTR6HTR2CHTR2ABRD4PTGDR2
SCHEMBL6086419 0.84 HTR2C (0.54) HTR6HTR2CHTR2ABRD4PTGDR2
SCHEMBL6086069 0.81 CCR2 (0.54) HTR6HTR2CHTR2ABRD4PTGDR2
SCHEMBL28101302 0.81 HTR6 (0.60) HTR6APPSNCABRD4BACE1
SCHEMBL6086525 0.80 CYP11B1 (0.48) HTR6APPSNCAHTR2CHTR2A
SCHEMBL4943583 0.80 HTR6 (0.58) HTR6APPSNCABRD4BACE1
SCHEMBL5134071 0.80 HTR6 (0.66) HTR6APPSNCABRD4BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110218206-B Bisindolylmaleimide derivative and preparation method and application thereof 中国海洋大学 2022-03-04 CN disclosed
CN-110526903-B Bisindolylmaleimide derivative and preparation method and application thereof 中国海洋大学 2021-12-10 CN disclosed
CN-110526903-A Bisindole maleimide derivative and its preparation method and application OCEAN UNIV CHINA 2019-12-03 CN disclosed
CN-110218206-A Bisindole maleimide derivative and its preparation method and application 中国海洋大学 2019-09-10 CN disclosed
CN-106083830-B Bisindolylmaleimide derivative and preparation method and application thereof 中国海洋大学 2019-07-12 CN disclosed
CN-106146475-B Bisindolylmaleimide derivative and preparation method and application thereof 中国海洋大学 2019-05-17 CN disclosed
CN-106146475-A Bisindolylmaleimide derivative and preparation method and application thereof 中国海洋大学 2016-11-23 CN disclosed
CN-106083830-A Bisindolylmaleimide derivative and preparation method and application thereof 中国海洋大学 2016-11-09 CN disclosed
US-4895958-A CHROMOGENS, IMAGES, PRESSURE SENSITIVE AND HEAT RESPONSIVE CARBONLESS DUPLICATING HILTON DAVIS CO. (US) 1990-01-23 US disclosed
US-4795736-A AMINOPHENYL PHENYLSULFONYL PROPENE/1-/ HILTON DAVIS CO. (US) 1989-01-03 US disclosed
US-4403791-A Carbonless duplicating and marking systems STERLING DRUG INC. (US) 1983-09-13 US disclosed
US-4377698-A 2,4 Bis(2-indolyl-3)-4-oxobutanoic acids STERLING DRUG INC. (US) 1983-03-22 US disclosed
US-4351768-A CARBONLESS, DUPLICATION, INDOLE DYES STERLING DRUG INC. (US) 1982-09-28 US disclosed
US-4322352-A Indolyl phthalide compounds STERLING DRUG INC. (US) 1982-03-30 US disclosed
US-4307018-A CHROMOGENS FOR COPYING SYSTEMS STERLING DRUG INC. (US) 1981-12-22 US disclosed
US-4275121-A Carbonless duplicating and marking systems utilizing indolyl-substituted furanone color formers STERLING DRUG INC. (US) 1981-06-23 US disclosed
US-4257954-A INDOLYL-PHENYLSULFONYL-PHENYL METHANE STERLING DRUG INC. (US) 1981-03-24 US disclosed
US-4251446-A COLOR PRECURSORS STERLING DRUG INC. (US) 1981-02-17 US disclosed
US-4189171-A PRESSURE SENSITIVE, THERMAL AND HECTOGRAPHIC SYSTEMS STERLING DRUG INC. (US) 1980-02-19 US disclosed
US-4075224-A 3,5-Bis (indolyl)-5-(indolyl)-2(5H)-furanones STERLING DRUG INC. (US) 1978-02-21 US disclosed