SCHEMBL5134071

SCHEMBL5134071

Nc1ccc2ccn(Cc3ccccc3)c2c1.Nc1ccc2ccn(Cc3ccccc3)c2c1

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.66
APP P05067 4/20 0.53
SNCA P37840 3/20 0.53
BRD4 O60885 3/20 0.50
BACE1 P56817 1/20 0.48
PLAU P00749 2/20 0.47
SLC2A1 P11166 1/20 0.45
NPC1 O15118 1/20 0.44
HSP90AA1 P07900 1/20 0.44
KMT2A Q03164 1/20 0.43
KDM4C Q9H3R0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL396279 1.00 HTR6 (0.66) HTR6APPSNCABRD4BACE1
SCHEMBL30241534 0.87 HTR6 (0.66) HTR6APPSNCAPLAUSLC2A1
SCHEMBL2769024 0.87 HTR6 (0.66) HTR6APPSNCAPLAUSLC2A1
SCHEMBL1122491 0.84 NOS1 (0.52) HTR6KMT2A
SCHEMBL916458 0.82 HTR6 (0.51) HTR6PLAUKMT2AKDM4C
SCHEMBL24414631 0.82 HTR6 (0.57) HTR6APPSNCABRD4BACE1
SCHEMBL28101302 0.81 HTR6 (0.60) HTR6APPSNCABRD4BACE1
SCHEMBL710269 0.81 HTR6 (0.50) HTR6APPSNCABRD4BACE1
SCHEMBL17602070 0.80 BACE1 (0.61) HTR6APPSNCABRD4BACE1
SCHEMBL4943583 0.80 HTR6 (0.58) HTR6APPSNCABRD4BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2489659-A1 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-08-22 EP disclosed
EP-1974212-A1 COMPOUNDS USEFUL IN CFTR ASSAYS AND METHODS THEREWITH Vertex Pharmaceuticals Incorporated (US) 2008-10-01 EP disclosed
WO-2007075946-A1 COMPOUNDS USEFUL IN CFTR ASSAYS AND METHODS THEREWITH VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-07-05 WO disclosed
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed