SCHEMBL10423366

SCHEMBL10423366

CN1CCC(Oc2c(F)c(F)c(F)c(F)c2F)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.39
CHRM2 P08172 2/20 0.37
CHRM1 P11229 2/20 0.37
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
CYP2D6 P10635 1/20 0.37
DRD1 P21728 1/20 0.37
SLC6A2 P23975 1/20 0.37
ADRA1A P35348 1/20 0.37
OPRM1 P35372 1/20 0.37
DRD3 P35462 1/20 0.37
SLC6A3 Q01959 1/20 0.37
KCNH2 Q12809 1/20 0.37
MAPK1 P28482 1/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 1/20 0.36
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM3 P20309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10424431 0.98 SMN1; SMN2 (0.41) HRH3SMN1; SMN2CHRM2CHRM1HTR1A
SCHEMBL10423406 0.79 HRH3 (0.47) HRH3SMN1; SMN2CHRM3
SCHEMBL20165826 0.78 SLC6A4 (0.32) CHRM4CHRM3
SCHEMBL9463735 0.76 SCD (0.30)
SCHEMBL10423361 0.76 HRH3 (0.34) HRH3
SCHEMBL10423372 0.76 ALOX15 (0.40) HRH3DRD3CHRM3
SCHEMBL9463387 0.76 IKBKB (0.40) SMN1; SMN2KMT2AMEN1
SCHEMBL10423401 0.76 CARM1 (0.58) HRH3
SCHEMBL10424979 0.76 CARM1 (0.35) HRH3SLC6A3KCNH2
SCHEMBL27092109 0.75 THRA (0.33) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4954511-A ALLEVIATING PAIN, TREATING DEPRESSION, CONVULSIONS AND HYPERTENSION HOECHST-ROUSSELL PHARMACEUTICALS INC. (US) 1990-09-04 US claimed
US-4954511-A ALLEVIATING PAIN, TREATING DEPRESSION, CONVULSIONS AND HYPERTENSION HOECHST-ROUSSELL PHARMACEUTICALS INC. (US) 1990-09-04 US disclosed
US-4914204-A ANALGESICS, ANTIDEPRESSANTS, ANTICONVULSANTS, HYPOTENSIVE AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1990-04-03 US disclosed
EP-0333027-A1 4-Pentafluorophenoxypiperidines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-09-20 EP disclosed