SCHEMBL10427019

SCHEMBL10427019

COc1cc2c(cc1OC)C(=O)C(CCC(=O)O)CC2

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.48
NQO2 P16083 1/20 0.46
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
CYP26A1 O43174 1/20 0.44
CYP24A1 Q07973 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27599825 0.91 ACHE (0.46) ACHENQO2MTNR1AMTNR1B
SCHEMBL10427888 0.88 ACHE (0.46) ACHENQO2MTNR1AMTNR1B
SCHEMBL10426976 0.86 ACHE (0.54) ACHE
SCHEMBL10700406 0.86 NQO2 (0.46) ACHENQO2MTNR1AMTNR1B
SCHEMBL4621209 0.82 CYP24A1 (0.65) ACHECYP26A1CYP24A1
SCHEMBL7171991 0.81 HDAC6 (0.51) ACHENQO2MTNR1AMTNR1B
SCHEMBL8535560 0.80 CYP19A1 (0.62) ACHEMTNR1AMTNR1B
SCHEMBL7249948 0.77 ACHE (0.64) ACHECYP26A1CYP24A1
SCHEMBL10427929 0.77 CDK8 (0.53) ACHE
SCHEMBL8531158 0.77 KMT2A (0.48) ACHENQO2MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0259782-B1 NAPHTHALENE AND INDANE DERIVATIVES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESSES FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-12-27 EP disclosed
EP-0259782-A1 Naphthalene and indane derivatives, medicaments containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1988-03-16 EP disclosed