SCHEMBL10427752

SCHEMBL10427752

O=c1c(Br)c(O)c2cccnc2n1-c1cccc(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.50
MAPT P10636 3/20 0.50
MEN1 O00255 2/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2C19 P33261 2/20 0.50
HPGD P15428 1/20 0.50
KDM4E B2RXH2 4/20 0.43
GAA P10253 1/20 0.43
FEN1 P39748 1/20 0.43
PDE4B Q07343 3/20 0.41
PDE4D Q08499 3/20 0.41
SLC22A12 Q96S37 1/20 0.40
PDE4A P27815 4/20 0.40
PDE4C Q08493 2/20 0.40
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALDH1A1 P00352 2/20 0.39
IDO1 P14902 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9715610 0.85 FEN1 (0.58) KMT2AMAPTCYP2C19HPGDKDM4E
SCHEMBL9267553 0.82 MAPT (0.47) KMT2AMAPTMEN1CYP1A2CYP2C19
SCHEMBL7272901 0.81 PDE4A (0.48) KMT2AMAPTMEN1CYP1A2CYP2C19
SCHEMBL9348307 0.80 CYP1A2 (0.46) KMT2AMAPTMEN1CYP1A2CYP2C19
SCHEMBL9348283 0.78 MAPT (0.46) KMT2AMAPTMEN1CYP1A2CYP2C19
SCHEMBL9799559 0.78 CYP1A2 (0.44) KMT2AMAPTMEN1CYP1A2CYP2C19
Water SCHEMBL10427748 0.78 MAPT (0.44) KMT2AMAPTMEN1CYP1A2CYP2C19
SCHEMBL10427749 0.77 MEN1 (0.42) KMT2AMAPTMEN1CYP1A2CYP2C19
Water SCHEMBL9715615 0.77 MAPT (0.42) KMT2AMAPTMEN1CYP1A2CYP2C19
SCHEMBL9535601 0.75 MAPT (0.50) KMT2AMAPTMEN1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4902693-A Anti-allergic esters, acetal ethers, thioethers and nitrogen substituted derivatives of bicyclic compounds SCHERING CORPORATION (US) 1990-02-20 US disclosed
US-4794116-A ANTIINFLAMMATORY AGENTS, CYTOPROTECTIVE AGENTS IN TREATMENT OF HYPERPROLIFERATIVE SKIN DISEASE SCHERING CORPORATION (US) 1988-12-27 US disclosed
US-4782067-A Anti-allergic composition containing zwitterionic bicyclic compounds SCHERING CORPORATION (US) 1988-11-01 US disclosed
EP-0232328-A1 ZWITTERIONIC BICYCLIC COMPOUNDS AND THEIR SALTS, SOLVATES, HYDRATES AND ESTERS. SCHERING CORP (US) 1987-08-19 EP disclosed
US-4684727-A Zwitterionic 1,8-naphthyridine and pyrazino[2,3-b]pyridine containing compounds useful as anti-allergic, anti-inflammatory and cycloprotective agents SCHERING CORPORATION (US) 1987-08-04 US disclosed
WO-1987000752-A2 ZWITTERIONIC BICYCLIC COMPOUNDS AND THEIR SALTS, SOLVATES, HYDRATES AND ESTERS SCHERING CORPORATION (US) 1987-02-12 WO disclosed