SCHEMBL9799559

SCHEMBL9799559

CC(O)Cc1c(O)c2cccnc2n(-c2cccc(Cl)c2)c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
CYP2C19 P33261 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 2/20 0.44
HPGD P15428 1/20 0.44
DRD1 P21728 1/20 0.41
DRD5 P21918 1/20 0.41
PDE4A P27815 6/20 0.40
PDE4B Q07343 4/20 0.40
PDE4C Q08493 4/20 0.40
PDE4D Q08499 4/20 0.40
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
KDM4E B2RXH2 3/20 0.39
SLC2A1 P11166 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10377267 0.88 KAT2B (0.42) MAPTPDE4APDE4BPDE4CPDE4D
SCHEMBL10377449 0.88 PDE4A (0.51) CYP1A2CYP2C19MAPTHPGDPDE4A
SCHEMBL9799463 0.88 KAT2B (0.45) MEN1KMT2AMAPTPDE4APDE4B
SCHEMBL9348283 0.81 MAPT (0.46) CYP1A2CYP2C19MEN1KMT2AMAPT
SCHEMBL9348307 0.80 CYP1A2 (0.46) CYP1A2CYP2C19MEN1KMT2AMAPT
SCHEMBL8803476 0.80 PDE4A (0.55) CYP1A2CYP2C19MAPTHPGDDRD1
SCHEMBL10427752 0.78 KMT2A (0.50) CYP1A2CYP2C19MEN1KMT2AMAPT
SCHEMBL9267553 0.78 MAPT (0.47) CYP1A2CYP2C19MEN1KMT2AMAPT
SCHEMBL7272901 0.75 PDE4A (0.48) CYP1A2CYP2C19MEN1KMT2AMAPT
SCHEMBL9215901 0.74 MAPT (0.44) CYP1A2CYP2C19MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4996212-A Antiinflammatory and anti-hyperproliferative compounds SCHERING CORPORATION (US) 1991-02-26 US disclosed
US-4859669-A Antiinflammatory and anti-hyperproliferative naphthyridin-4-ones SCHERING CORPORATION (US) 1989-08-22 US disclosed