SCHEMBL10429366

SCHEMBL10429366

COc1ccc(-c2nccc(C#N)c2N)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.54
ADORA2A P29274 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.48
DYRK1A Q13627 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
KDM4E B2RXH2 4/20 0.46
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 2/20 0.46
HPGD P15428 1/20 0.45
MYC P01106 1/20 0.44
WDR5 P61964 1/20 0.44
CSNK2A1 P68400 1/20 0.42
CDK1 P06493 1/20 0.42
KDR P35968 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1003068 0.79 DYRK1A (0.53) ADORA1ADORA2ASMN1; SMN2DYRK1ANPC1
SCHEMBL10429370 0.79 ADORA1 (0.54) ADORA1ADORA2AKDM4EKMT2AALDH1A1
SCHEMBL16879478 0.78 ALDH1A1 (0.59) ADORA1ADORA2ASMN1; SMN2NPC1RAB9A
SCHEMBL16891621 0.75 ADORA1 (0.66) ADORA1ADORA2ANPC1RAB9AKDM4E
SCHEMBL16739956 0.74 ADORA2A (0.50) ADORA1ADORA2ASMN1; SMN2KDM4EKMT2A
SCHEMBL7689092 0.72 POLB (0.49) ADORA1ADORA2ASMN1; SMN2NPC1RAB9A
SCHEMBL18447982 0.72 TDP1 (0.61) ADORA1SMN1; SMN2DYRK1ANPC1RAB9A
SCHEMBL20522349 0.72 KDM4E (0.54) ADORA1ADORA2ADYRK1ANPC1RAB9A
SCHEMBL30610423 0.72 KDM4E (0.54) ADORA1ADORA2ADYRK1ANPC1RAB9A
SCHEMBL10429365 0.72 KDM4E (0.52) DYRK1AKDM4EKMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4920119-A XANTHINE OXIDASE INHIBITORS; CONTROL OR PREVENTION OF GOUT OR ISCHEMIA HOFFMANN-LA ROCHE INC. (US) 1990-04-24 US disclosed
EP-0274654-A2 1,2,3-Triazin-4(3H)-one derivatives, process for their preparation and medicaments containing them F. HOFFMANN-LA ROCHE AG (CH) 1988-07-20 EP disclosed