SCHEMBL10434205

SCHEMBL10434205

CC(C)c1nc(-c2ccccc2)nc(-c2ccc(F)cc2)c1C=CC=O

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 7/20 0.57
DPP4 P27487 1/20 0.41
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.39
PDE6D O43924 1/20 0.39
NR1I2 O75469 1/20 0.39
PDE4D Q08499 1/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
GCGR P47871 1/20 0.38
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ABCC3 O15438 1/20 0.36
ABCC4 O15439 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10433924 1.00 HMGCR (0.57) HMGCRDPP4ALDH1A1CYP3A4PDE6D
SCHEMBL9788409 0.91 HMGCR (0.51) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL9562922 0.88 HMGCR (0.56) HMGCRDPP4ALDH1A1CYP3A4PDE6D
SCHEMBL9562755 0.85 HMGCR (0.56) HMGCRDPP4ALDH1A1CYP3A4PDE6D
SCHEMBL9562749 0.85 HMGCR (0.56) HMGCRDPP4ALDH1A1CYP3A4PDE6D
SCHEMBL9788395 0.85 DPP4 (0.45) HMGCRDPP4ALDH1A1PDE4DHTR2A
SCHEMBL9521683 0.83 HMGCR (0.53) HMGCRDPP4ALDH1A1CYP3A4PDE6D
SCHEMBL8846369 0.83 HMGCR (0.53) HMGCRDPP4ALDH1A1CYP3A4HTR2A
SCHEMBL10129259 0.80 HMGCR (0.48) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL17875116 0.80 ADORA1 (0.41) HMGCRALDH1A1CYP3A4PDE6DNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0367895-A1 Pyrimidinyl-substituted hydroxyacids, lactones and esters and pharmaceutical compositions containing them SANDOZ AG (CH) 1990-05-16 EP disclosed