SCHEMBL10436780

SCHEMBL10436780

FC(F)(F)c1ccc2nccc(-c3ccccc3)c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.57
CCNC P24863 1/20 0.53
CDK8 P49336 1/20 0.53
GRM4 Q14833 1/20 0.53
MAPK14 Q16539 2/20 0.50
TGFBR1 P36897 1/20 0.50
SLC22A12 Q96S37 2/20 0.47
TOP1 P11387 1/20 0.47
NPBWR1 P48145 1/20 0.46
PTGDR2 Q9Y5Y4 2/20 0.45
GAK O14976 2/20 0.44
DGAT1 O75907 1/20 0.43
KCNH2 Q12809 1/20 0.43
RIPK2 O43353 2/20 0.43
DHODH Q02127 1/20 0.43
KDR P35968 1/20 0.43
KIF11 P52732 1/20 0.43
EPHB6 O15197 1/20 0.42
ABL1 P00519 1/20 0.42
LCK P06239 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28170035 0.88 GRM4 (0.67) PIK3CACCNCCDK8GRM4MAPK14
SCHEMBL31222481 0.81 TGFBR1 (0.52) PIK3CAGRM4MAPK14TGFBR1TOP1
SCHEMBL28118653 0.79 TOP1 (0.58) TOP1NPBWR1DGAT1KCNH2DHODH
SCHEMBL9709110 0.78 PIK3CA (0.87) PIK3CACDK8KDR
SCHEMBL14349100 0.78 P2RX1 (0.50)
SCHEMBL11831483 0.77 NPBWR1 (0.48) TOP1NPBWR1DGAT1KCNH2DHODH
SCHEMBL12277881 0.76 PIK3CA (0.62) PIK3CACCNCCDK8SLC22A12KDR
SCHEMBL30440259 0.76 PIK3CA (0.62) PIK3CACCNCCDK8SLC22A12KDR
SCHEMBL9806116 0.76 PIK3CA (0.62) PIK3CACDK8SLC22A12KDR
SCHEMBL8956040 0.76 PIK3CA (0.62) PIK3CACCNCCDK8GRM4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0354994-A2 Quinoline derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-02-21 EP disclosed