SCHEMBL10437652

SCHEMBL10437652

c1ccc(COc2ccc(N3CCc4ccccc4CC3)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 9/20 0.58
PRMT5 O14744 2/20 0.54
WDR77 Q9BQA1 2/20 0.54
RAB9A P51151 2/20 0.51
NPC1 O15118 1/20 0.51
TP53 P04637 1/20 0.51
CYP2D6 P10635 3/20 0.51
HRH1 P35367 1/20 0.51
MAPT P10636 3/20 0.50
LMNA P02545 2/20 0.50
LTA4H P09960 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HTT P42858 1/20 0.50
CYP1A2 P05177 1/20 0.50
PTGS1 P23219 1/20 0.50
SLC6A2 P23975 1/20 0.50
CYP2C19 P33261 1/20 0.50
PTGS2 P35354 1/20 0.50
SLC6A3 Q01959 1/20 0.50
HIF1A Q16665 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3089244 0.87 HRH3 (0.74) HRH3CYP2D6HRH1GRIN1GRIN2B
SCHEMBL735870 0.86 MAPT (0.52) HRH3RAB9ANPC1MAPTLMNA
SCHEMBL16046663 0.85 LTA4H (0.62) HRH3RAB9ANPC1TP53MAPT
SCHEMBL13202898 0.84 RAB9A (0.67) HRH3PRMT5RAB9ANPC1TP53
SCHEMBL9047395 0.84 LTA4H (0.60) HRH3RAB9ANPC1LMNALTA4H
SCHEMBL738629 0.84 MAOB (0.54) HRH3RAB9ANPC1TP53MAPT
SCHEMBL2342568 0.83 LMNA (0.51) HRH3RAB9ANPC1TP53MAPT
SCHEMBL13279833 0.82 GSTP1 (0.52) RAB9ANPC1MAPTLMNALTA4H
SCHEMBL7891469 0.82 MAPT (0.49) HRH3RAB9ANPC1MAPTLMNA
SCHEMBL335477 0.81 LTA4H (0.64) PRMT5MAPTLMNALTA4HALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0380355-A2 Carbamates of 6-chloro-7,8-dihydroxy-1-(4'-Hydroxyphenyl)-2,3,4,5-tetra-hydro-1H-3-benzazepine as prodrugs SMITHKLINE BEECHAM CORPORATION (US) 1990-08-01 EP disclosed