SCHEMBL10440314

SCHEMBL10440314

Cc1ccc(N2C(=O)[C@@H]3CCCCN3C2=O)c(F)c1O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.43
POLB P06746 1/20 0.40
ALDH1A1 P00352 3/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 3/20 0.37
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
THRB P10828 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10440318 0.78 AR (0.45) ARPOLBALDH1A1HTTKMT2A
SCHEMBL11038098 0.72 AR (0.52) ARPOLBALDH1A1KMT2ASMN1; SMN2
SCHEMBL10935874 0.71 AR (0.45) ARALDH1A1KMT2ASMN1; SMN2
SCHEMBL9664391 0.71 AR (0.45) ARPOLBALDH1A1KMT2ASMN1; SMN2
SCHEMBL13879455 0.69 KDM4E (0.56) ARPOLBALDH1A1HTTKMT2A
SCHEMBL13879486 0.69 ALDH1A1 (0.56) ARPOLBALDH1A1HTTKMT2A
SCHEMBL10463025 0.68 AR (0.40) ARPOLBALDH1A1KMT2AKDM4E
SCHEMBL1514017 0.68 AR (0.43) ARPOLBALDH1A1HTTKMT2A
SCHEMBL9382971 0.68 AR (0.42) ARALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL1513976 0.68 ALDH1A1 (0.52) ARPOLBALDH1A1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0363585-A1 N-aryl nitrogen heterocycles BAYER AG (DE) 1990-04-18 EP disclosed