SCHEMBL10440323

SCHEMBL10440323

COC(=O)C(C)Oc1cc(N)ccc1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH2 P05091 1/20 0.44
F9 P00740 1/20 0.43
PLAU P00749 1/20 0.43
ALDH1A1 P00352 5/20 0.42
TSHR P16473 5/20 0.41
HPGD P15428 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPK1 P28482 1/20 0.41
TAS1R3 Q7RTX0 2/20 0.40
TAS1R1 Q7RTX1 2/20 0.40
GAA P10253 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALOX5 P09917 1/20 0.40
RECQL P46063 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CASP1 P29466 2/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24419010 0.85 TSHR (0.48) ALDH2F9PLAUALDH1A1TSHR
SCHEMBL22542376 0.85 ALDH2 (0.55) ALDH2F9PLAUALDH1A1TSHR
SCHEMBL11689564 0.85 TDP1 (0.56) ALDH1A1TSHRHPGDHSD17B10KDM4E
SCHEMBL22542369 0.81 ALDH2 (0.51) ALDH2F9PLAUALDH1A1TSHR
SCHEMBL9823852 0.79 GAA (0.47) ALDH2F9PLAUALDH1A1HPGD
SCHEMBL4017962 0.78 ALDH1A1 (0.50) ALDH1A1TSHRHPGDHSD17B10KDM4E
SCHEMBL21415510 0.78 HPGD (0.56) ALDH2F9PLAUALDH1A1TSHR
SCHEMBL20097882 0.78 HPGD (0.56) ALDH2F9PLAUALDH1A1TSHR
SCHEMBL10051619 0.78 TAS1R3 (0.40) ALDH1A1TSHRTAS1R3TAS1R1GAA
SCHEMBL11691601 0.78 CASP1 (0.45) ALDH1A1TSHRKDM4EMAPK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0363585-A1 N-aryl nitrogen heterocycles BAYER AG (DE) 1990-04-18 EP disclosed