SCHEMBL1044324

SCHEMBL1044324

C=CCC(=C)C(=O)OC(=O)OC(=O)C(=C)CC=C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL244290 0.90 ALDH1A1 (0.31)
SCHEMBL1049922 0.84 ALOX15 (0.31)
SCHEMBL244291 0.82 TSHR (0.35)
SCHEMBL28066529 0.82 HSD17B10 (0.42)
SCHEMBL10434293 0.80 TSHR (0.34)
SCHEMBL44693 0.78
SCHEMBL8166432 0.76
SCHEMBL15690510 0.76
SCHEMBL1950793 0.76
SCHEMBL2405615 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2729457-B1 METHOD FOR MAKING A POLYMER, A POLYMER ARTICLE, A BIODEVICE, AND CYCLIC CARBONATE SSENS B V (NL) 2016-11-02 EP claimed
EP-2456764-B1 A METHOD OF MAKING A POLYMER PREFERABLY AN (ALKYL)ACRYLOYL POLYCARBONATE, THE POLYMER AND (ALKYL)ACRYLOYL POLYCARBONATE OBTAINED, AND A BIODEVICE COMPRISING SAME SSENS B V (NL) 2016-03-30 EP claimed
US-8927196-B2 Method of making an (alkyl)acryloyl polycarbonate SSENS B.V. (NL) 2015-01-06 US claimed
US-20120294845-A1 METHOD OF MAKING A POLYMER PREFERABLY AN (ALKYL) ACRYLOYL POLYCARBONATE, THE POLYMER AND (ALKYL) ACRYLOYL POLYCARBONATE OBTAINED, AND A BIODEVICE COMPRISING SAME SSENS B.V. (NL) 2012-11-22 US claimed
EP-2456764-A1 A METHOD OF MAKING A POLYMER PREFERABLY AN (ALKYL)ACRYLOYL POLYCARBONATE, THE POLYMER AND (ALKYL)ACRYLOYL POLYCARBONATE OBTAINED, AND A BIODEVICE COMPRISING SAME Ssens B.V. (NL) 2012-05-30 EP claimed
EP-2456764-B1 A METHOD OF MAKING A POLYMER PREFERABLY AN (ALKYL)ACRYLOYL POLYCARBONATE, THE POLYMER AND (ALKYL)ACRYLOYL POLYCARBONATE OBTAINED, AND A BIODEVICE COMPRISING SAME SSENS B V (NL) 2016-03-30 EP disclosed
US-8927196-B2 Method of making an (alkyl)acryloyl polycarbonate SSENS B.V. (NL) 2015-01-06 US disclosed
US-8927196-B2 Method of making an (alkyl)acryloyl polycarbonate SSENS B.V. (NL) 2015-01-06 US disclosed
EP-2729457-A1 METHOD FOR MAKING A POLYMER, A POLYMER ARTICLE, A BIODEVICE, AND CYCLIC CARBONATE Ssens B.V. (NL) 2014-05-14 EP disclosed
WO-2013004296-A1 METHOD FOR MAKING A POLYMER, A POLYMER ARTICLE, A BIODEVICE, AND CYCLIC CARBONATE SSENS B.V. (NL) 2013-01-10 WO disclosed
US-20120294845-A1 METHOD OF MAKING A POLYMER PREFERABLY AN (ALKYL) ACRYLOYL POLYCARBONATE, THE POLYMER AND (ALKYL) ACRYLOYL POLYCARBONATE OBTAINED, AND A BIODEVICE COMPRISING SAME SSENS B.V. (NL) 2012-11-22 US disclosed
US-20120294845-A1 METHOD OF MAKING A POLYMER PREFERABLY AN (ALKYL) ACRYLOYL POLYCARBONATE, THE POLYMER AND (ALKYL) ACRYLOYL POLYCARBONATE OBTAINED, AND A BIODEVICE COMPRISING SAME SSENS B.V. (NL) 2012-11-22 US disclosed
CN-102712616-A A method of making a polymer preferably an (alkyl) acryloyl polycarbonate, the polymer and (alkyl)acryloyl polycarbonate obtained, and a biodevice comprising same SSENS B V 2012-10-03 CN disclosed
EP-2456764-A1 A METHOD OF MAKING A POLYMER PREFERABLY AN (ALKYL)ACRYLOYL POLYCARBONATE, THE POLYMER AND (ALKYL)ACRYLOYL POLYCARBONATE OBTAINED, AND A BIODEVICE COMPRISING SAME Ssens B.V. (NL) 2012-05-30 EP disclosed
EP-2456764-A1 A METHOD OF MAKING A POLYMER PREFERABLY AN (ALKYL)ACRYLOYL POLYCARBONATE, THE POLYMER AND (ALKYL)ACRYLOYL POLYCARBONATE OBTAINED, AND A BIODEVICE COMPRISING SAME Ssens B.V. (NL) 2012-05-30 EP disclosed
WO-2011009478-A1 A METHOD OF MAKING A POLYMER PREFERABLY AN (ALKYL)ACRYLOYL POLYCARBONATE, THE POLYMER AND (ALKYL)ACRYLOYL POLYCARBONATE OBTAINED, AND A BIODEVICE COMPRISING SAME SSENS B.V. (NL) 2011-01-27 WO disclosed
WO-2011009478-A1 A METHOD OF MAKING A POLYMER PREFERABLY AN (ALKYL)ACRYLOYL POLYCARBONATE, THE POLYMER AND (ALKYL)ACRYLOYL POLYCARBONATE OBTAINED, AND A BIODEVICE COMPRISING SAME SSENS B.V. (NL) 2011-01-27 WO disclosed