SCHEMBL10447258

SCHEMBL10447258

O=C(c1ccccc1F)C1CCN(CCc2ccccc2)CC1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 8/20 0.69
HTR2C P28335 3/20 0.59
HTR7 P34969 3/20 0.59
HTR6 P50406 3/20 0.59
OPRM1 P35372 2/20 0.58
KDM4E B2RXH2 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
GRM2 Q14416 2/20 0.57
KCNH2 Q12809 1/20 0.53
SIGMAR1 Q99720 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10164227 0.86 KMT2A (0.59) HTR2AHTR2CKDM4ESIGMAR1
SCHEMBL7839803 0.82 HTR2A (1.00) HTR2AHTR2CHTR7HTR6OPRM1
SCHEMBL1582470 0.82 HTR2A (0.87) HTR2AHTR2CHTR7HTR6KDM4E
Hydrochloric Acid SCHEMBL7828801 0.81 HTR2A (0.97) HTR2AHTR2CHTR7HTR6OPRM1
SCHEMBL10366605 0.81 HSD11B1 (0.51) HTR2AHTR2CHTR7HTR6GRM2
Hydrochloric Acid SCHEMBL7418228 0.81 HTR2A (0.85) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL27300983 0.80 HTR2A (0.75) HTR2AHTR2COPRM1KDM4ECYP1A2
SCHEMBL1519356 0.80 HTR2A (0.75) HTR2AOPRM1SIGMAR1
Hydrochloric Acid SCHEMBL10365798 0.80 HSD11B1 (0.50) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL6661943 0.79 HSD11B1 (0.55) HTR7SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0360275-A2 Imidazole antiarrhythmics MERRELL DOW PHARMACEUTICALS INC. (US) 1990-03-28 EP disclosed