SCHEMBL10448952

SCHEMBL10448952

COc1ccc(S(=O)(=O)NN(C)S(=O)(=O)c2ccc(Br)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.57
EGFR P00533 1/20 0.51
ERBB2 P04626 1/20 0.51
POLB P06746 1/20 0.50
MMP1 P03956 2/20 0.49
MMP9 P14780 2/20 0.49
MMP13 P45452 2/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
MMP2 P08253 1/20 0.49
MMP8 P22894 1/20 0.49
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
FFAR4 Q5NUL3 3/20 0.47
ADAM17 P78536 1/20 0.45
PKM P14618 2/20 0.45
KEAP1 Q14145 2/20 0.44
TP53 P04637 1/20 0.44
THRB P10828 1/20 0.44
CYP19A1 P11511 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10869544 1.00 IDO1 (0.57) IDO1EGFRERBB2POLBMMP1
SCHEMBL10620967 0.92 CA1 (0.56) MMP1MMP9MMP13CA1CA2
SCHEMBL10449067 0.89 MMP2 (0.50) IDO1MMP1MMP9MMP13CA1
SCHEMBL10449123 0.87 ALDH1A1 (0.55) EGFRPOLBMMP1MMP9MMP13
SCHEMBL10448918 0.85 ALDH1A1 (0.52) EGFRERBB2MMP1MMP9MMP13
SCHEMBL10448907 0.85 ALDH1A1 (0.52) EGFRERBB2MMP1MMP9MMP13
SCHEMBL10449124 0.83 IDO1 (0.49) IDO1EGFRERBB2MMP1MMP9
SCHEMBL10448742 0.83 EGFR (0.48) IDO1EGFRERBB2MMP1MMP9
SCHEMBL10449154 0.83 EGFR (0.48) IDO1EGFRERBB2MMP1MMP9
SCHEMBL10449155 0.82 TSHR (0.49) IDO1EGFRERBB2MMP1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4892887-A ANTITUMOR YALE UNIVERSITY (US) 1990-01-09 US disclosed
EP-0185387-B1 NOVEL, N,N'BIS(SULFONYL) HYDRAZINES HAVING ANTINEOPLASTIC ACTIVITY YALE UNIVERSITY (US) 1988-12-14 EP disclosed
US-4684747-A ANTITUMOR, ALKYLATING AGENTS YALE UNIVERSITY (US) 1987-08-04 US disclosed