SCHEMBL10449124

SCHEMBL10449124

CN(NS(=O)(=O)c1ccccc1)S(=O)(=O)c1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.49
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 2/20 0.46
HTT P42858 2/20 0.46
ALDH1A1 P00352 1/20 0.46
RECQL P46063 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
MMP1 P03956 1/20 0.44
MMP2 P08253 1/20 0.44
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
MMP13 P45452 1/20 0.44
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
RAB9A P51151 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
NAT1 P18440 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10449067 0.93 MMP2 (0.50) IDO1MEN1KMT2ALMNAHTT
SCHEMBL10448678 0.90 BCAT1 (0.47) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL10448742 0.87 EGFR (0.48) IDO1MEN1KMT2ALMNAALDH1A1
SCHEMBL10449154 0.87 EGFR (0.48) IDO1MEN1KMT2ALMNAALDH1A1
SCHEMBL10449155 0.86 TSHR (0.49) IDO1ALDH1A1CA1CA2MMP1
SCHEMBL10871212 0.86 TSHR (0.49) IDO1ALDH1A1CA1CA2MMP1
SCHEMBL10448709 0.85 CA12 (0.56) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL10448943 0.84 ALDH1A1 (0.50) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL10449126 0.84 L3MBTL1 (0.49) MEN1KMT2ALMNAHTTALDH1A1
SCHEMBL10620308 0.84 L3MBTL1 (0.53) MEN1KMT2ALMNAHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4892887-A ANTITUMOR YALE UNIVERSITY (US) 1990-01-09 US disclosed
EP-0185387-B1 NOVEL, N,N'BIS(SULFONYL) HYDRAZINES HAVING ANTINEOPLASTIC ACTIVITY YALE UNIVERSITY (US) 1988-12-14 EP disclosed
US-4684747-A ANTITUMOR, ALKYLATING AGENTS YALE UNIVERSITY (US) 1987-08-04 US disclosed
EP-0185387-A1 Novel, N,N'bis(sulfonyl) hydrazines having antineoplastic activity YALE UNIVERSITY (US) 1986-06-25 EP disclosed