SCHEMBL10453073

SCHEMBL10453073

O=P(Cl)(Cl)CCCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
HDAC3 O15379 1/20 0.47
MAPK1 P28482 1/20 0.47
ADRA1A P35348 1/20 0.47
HDAC4 P56524 1/20 0.47
SLC6A3 Q01959 1/20 0.47
HDAC1 Q13547 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
S1PR2 O95136 2/20 0.46
S1PR4 O95977 2/20 0.46
S1PR1 P21453 2/20 0.46
S1PR3 Q99500 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8729220 0.94 TSHR (0.55) TSHRHDAC3MAPK1ADRA1AHDAC4
SCHEMBL6824408 0.86 TSHR (0.55) TSHRSMN1; SMN2POLBHTR2ACETP
SCHEMBL217735 0.79 MAOA (0.50) TSHRHDAC1SMN1; SMN2MAOAMAOB
SCHEMBL4406117 0.78 S1PR2 (0.69) TSHRHDAC3MAPK1ADRA1AHDAC4
SCHEMBL7434180 0.78 TSHR (0.61) TSHRHDAC3MAPK1ADRA1AHDAC4
SCHEMBL7265672 0.77 TSHR (0.55) TSHRSMN1; SMN2POLBHTR2ACETP
SCHEMBL28529985 0.77 TSHR (0.50) TSHRHDAC3MAPK1ADRA1AHDAC4
Zinc Ion SCHEMBL28535948 0.77 TSHR (0.50) TSHRHDAC3MAPK1ADRA1AHDAC4
SCHEMBL8641479 0.75 TSHR (0.58) TSHRHDAC3MAPK1ADRA1AHDAC4
SCHEMBL11775231 0.74 TSHR (0.62) TSHRMAPK1S1PR2S1PR4S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4900860-A Process for preparing phosphonyloxyacyl amino acids E. R. SQUIBB & SONS, INC. (US) 1990-02-13 US disclosed
US-4885380-A REACTING PHOSPHONIC ACID DICHLORIDE WITH ALPHA-HYDROXY ACID TO FORM CYCLIC MIXED ANHYDRIDE; REACTING WITH AMINO ACID THOTTATHIL JOHN K (US) 1989-12-05 US disclosed
EP-0237264-A2 Process for preparing phosphonyloxyacyl amino acids and derivates thereof E.R. Squibb & Sons, Inc. (US) 1987-09-16 EP disclosed