SCHEMBL10464779

SCHEMBL10464779

COC(=O)c1ccc(COc2ccc(C=O)cc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.73
RAB9A P51151 6/20 0.73
ALDH1A1 P00352 3/20 0.68
MAPT P10636 5/20 0.68
SMN1; SMN2 Q16637 4/20 0.68
MEN1 O00255 2/20 0.68
KMT2A Q03164 2/20 0.68
PKM P14618 1/20 0.60
KDM4E B2RXH2 2/20 0.59
CTSK P43235 1/20 0.57
LMNA P02545 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
PTPN1 P18031 2/20 0.55
POLB P06746 1/20 0.54
RXRA P19793 1/20 0.54
RXRB P28702 1/20 0.54
PSEN1 P49768 1/20 0.54
PSEN2 P49810 1/20 0.54
APH1B Q8WW43 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18259961 1.00 NPC1 (0.73) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL11350421 0.89 RAB9A (0.82) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL10236929 0.89 RAB9A (0.82) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL15565832 0.87 RAB9A (0.69) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL210094 0.86 MAPT (0.77) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL9128908 0.86 RAB9A (0.55) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL874405 0.85 MAOB (0.69) RAB9AALDH1A1SMN1; SMN2L3MBTL1HTT
SCHEMBL3729907 0.84 NPC1 (0.75) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL12086470 0.84 RAB9A (0.80) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL31482044 0.84 MRGPRX4 (0.56) NPC1RAB9AALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025080049-A1 COMPOUND FOR INHIBITING ATX, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION FOR USE IN PREVENTING OR TREATING ATX ACTIVITY-RELATED DISEASES CONTAINING SAME AS ACTIVE INGREDIENT 한국화학연구원 2025-04-17 WO disclosed
US-20250011285-A1 CYP11A1 INHIBITORS ORION CORPORATION (FI) 2025-01-09 US disclosed
EP-3152204-B1 CARBAMATE DERIVATIVES WHICH ARE BOTH PHOSPHODIESTERASE 4 (PDE4) ENZYME INHIBITORS AND MUSCARINIC M3 RECEPTOR ANTAGONISTS CHIESI FARM SPA (IT) 2018-03-28 EP disclosed
EP-2928880-B1 PHENYLETHYLPYRIDINE DERIVATIVES AS PDE4-INHIBITORS AND MUSCARINIC RECEPTOR ANTAGONISTS CHIESI FARM SPA (IT) 2018-02-14 EP disclosed
EP-2928880-B1 PHENYLETHYLPYRIDINE DERIVATIVES AS PDE4-INHIBITORS AND MUSCARINIC RECEPTOR ANTAGONISTS CHIESI FARM SPA (IT) 2018-02-14 EP disclosed
CN-104837828-B It is used as the phenylethyl pyridine derivate of PDE4 inhibitor 奇斯药制品公司 2017-07-18 CN disclosed
EP-2882740-B1 IAP ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2017-03-01 EP disclosed
US-9453048-B2 IAP antagonists BRISTOL-MYERS SQUIBB COMPANY (US) 2016-09-27 US disclosed
US-9326976-B2 Carbamate derivatives CHIESI FARMACEUTICI S.P.A. (IT) 2016-05-03 US disclosed
US-9326976-B2 Carbamate derivatives CHIESI FARMACEUTICI S.P.A. (IT) 2016-05-03 US disclosed
US-20140121213-A1 VOLTAGE-GATED SODIUM CHANNEL BLOCKERS GLAXO GROUP LIMITED (GB) 2014-05-01 US disclosed
WO-2014025759-A1 IAP ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2014-02-13 WO disclosed
US-20130023541-A1 VOLTAGE-GATED SODIUM CHANNEL BLOCKERS GLAXO GROUP LIMITED 2013-01-24 US disclosed
US-20130023541-A1 VOLTAGE-GATED SODIUM CHANNEL BLOCKERS GLAXO GROUP LIMITED 2013-01-24 US disclosed
US-20100216762-A1 Agonists and Antagonists of the S1P5 Receptor, and Methods of Use Thereof ABBOTT LABORATORIES (US) 2010-08-26 US disclosed
US-20100216762-A1 Agonists and Antagonists of the S1P5 Receptor, and Methods of Use Thereof ABBOTT LABORATORIES (US) 2010-08-26 US disclosed
EP-0397746-A1 CONDENSATION POLYMERS CONTAINING METHINE ULTRAVIOLET RADIATION-ABSORBING RESIDUES AND SHAPED ARTICLES PRODUCED THEREFROM EASTMAN KODAK COMPANY (US) 1990-11-22 EP disclosed
EP-0326287-A2 Condensation polymers containing methine ultraviolet radiation-absorbing residues and shaped articles produced therefrom EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1989-08-02 EP disclosed
WO-1989006663-A1 CONDENSATION POLYMERS CONTAINING METHINE ULTRAVIOLET RADIATION-ABSORBING RESIDUES AND SHAPED ARTICLES PRODUCED THEREFROM EASTMAN KODAK COMPANY (US) 1989-07-27 WO disclosed
US-4845187-A POLYESTERS EASTMAN KODAK COMPANY (US) 1989-07-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250011285-A1 CYP11A1 INHIBITORS CYP11B1, CYP19A1, CYP11B2 NPC1 695/4885RAB9A 2559/4885ALDH1A1 188/4885
US-20130023541-A1 VOLTAGE-GATED SODIUM CHANNEL BLOCKERS KCNB1, KCNB2, SCNN1B NPC1 670/4885RAB9A 1723/4885ALDH1A1 2656/4885
US-20140121213-A1 VOLTAGE-GATED SODIUM CHANNEL BLOCKERS KCNB1, SCNN1B, TRPV1 NPC1 620/4885RAB9A 2020/4885ALDH1A1 2495/4885
US-20100216762-A1 Agonists and Antagonists of the S1P5 Receptor, and Methods of Use Thereof S1PR5, LPAR5, S1PR1 NPC1 965/4885RAB9A 2255/4885ALDH1A1 1328/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.