SCHEMBL10467576

SCHEMBL10467576

O=C(O)/C=C/C1CC1(c1ccc(F)cc1)c1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 12/20 0.40
CCR2 P41597 1/20 0.38
PTGS2 P35354 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
MAOB P27338 2/20 0.37
MAOA P21397 1/20 0.37
GRIN2B Q13224 1/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10468097 1.00 HSD11B1 (0.40) HSD11B1CCR2PTGS2MEN1KMT2A
SCHEMBL10468088 1.00 HSD11B1 (0.40) HSD11B1CCR2PTGS2MEN1KMT2A
SCHEMBL10470144 1.00 HSD11B1 (0.40) HSD11B1CCR2PTGS2MEN1KMT2A
SCHEMBL10467434 0.85 LMNA (0.41) CCR2MEN1KMT2AALDH1A1LMNA
SCHEMBL10467989 0.85 LMNA (0.41) CCR2MEN1KMT2AALDH1A1LMNA
SCHEMBL10467452 0.85 LMNA (0.41) CCR2MEN1KMT2AALDH1A1LMNA
SCHEMBL10467712 0.85 LMNA (0.41) CCR2MEN1KMT2AALDH1A1LMNA
SCHEMBL10467453 0.85 LMNA (0.41) CCR2MEN1KMT2AALDH1A1LMNA
SCHEMBL10467674 0.85 LMNA (0.41) CCR2MEN1KMT2AALDH1A1LMNA
SCHEMBL10467987 0.85 LMNA (0.41) CCR2MEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4927826-A Cycloproylpropenamides useful as platelet activing factor (PAF) antagonists HOFFMAN-LA ROCHE INC. (US) 1990-05-22 US disclosed
US-4786646-A PLATELET ACTIVATING FACTOR ANTAGONISTS HOFFMANN-LA ROCHE INC. (US) 1988-11-22 US disclosed