SCHEMBL10472252

SCHEMBL10472252

O=C(NN1C(=O)Cc2ccccc21)c1ccccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.44
PTGS2 P35354 2/20 0.43
GAA P10253 2/20 0.43
NAMPT P43490 1/20 0.43
KDM4E B2RXH2 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
NOTUM Q6P988 1/20 0.42
TLR7 Q9NYK1 1/20 0.42
RAB9A P51151 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GRM5 P41594 1/20 0.41
NPC1 O15118 3/20 0.40
PKM P14618 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21099292 0.80 GRM4 (0.53) GRM4PTGS2GAAKDM4EKMT2A
SCHEMBL10472164 0.80 LMNA (0.57) GAAKDM4EKMT2ATDP1NOTUM
SCHEMBL7717408 0.79 MEN1 (0.51) GAAKDM4EKMT2ANOTUMSMN1; SMN2
SCHEMBL7476038 0.75 NOTUM (0.58) GAAKDM4EKMT2ATDP1NOTUM
SCHEMBL8812148 0.74 HPGD (0.41) GAAKDM4EKMT2ANOTUMRAB9A
SCHEMBL25215843 0.74 LMNA (0.60) GRM4PTGS2KDM4EKMT2ATLR7
SCHEMBL1290437 0.74 HPGD (0.44) KDM4EKMT2ATDP1NOTUM
SCHEMBL5624766 0.70 L3MBTL1 (0.40) KDM4ENOTUMSMN1; SMN2L3MBTL1PKM
SCHEMBL7471354 0.69 CYP2C19 (0.57) GAANAMPTKMT2ANOTUMRAB9A
SCHEMBL30761577 0.69 CNR1 (0.58) PTGS2GAAKDM4EKMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed