SCHEMBL10474113

SCHEMBL10474113

CCCCCCCCCCCc1cc(N)cc(OC)c1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.63
CYP19A1 P11511 1/20 0.50
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
GPR84 Q9NQS5 1/20 0.46
FUT7 Q11130 1/20 0.46
CNR1 P21554 9/20 0.45
CNR2 P34972 9/20 0.45
CYP3A4 P08684 1/20 0.43
HTR2A P28223 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15285314 0.93 PTGS2 (0.57) PTGS2CYP19A1CA1CA2CA9
SCHEMBL11089326 0.91 PTGS2 (0.54) PTGS2CYP19A1CA1CA2CA9
SCHEMBL18586439 0.87 PTGS2 (0.73) PTGS2CYP19A1CA1CA2CA9
SCHEMBL31185907 0.87 PTGS2 (0.73) PTGS2CYP19A1CA1CA2CA9
SCHEMBL31185803 0.87 PTGS2 (0.73) PTGS2CYP19A1CA1CA2CA9
SCHEMBL31185832 0.87 PTGS2 (0.73) PTGS2CYP19A1CA1CA2CA9
SCHEMBL20098971 0.85 CYP19A1 (0.56) PTGS2CYP19A1CYP3A4
SCHEMBL30380963 0.85 CYP19A1 (0.56) PTGS2CYP19A1CYP3A4
SCHEMBL1171756 0.85 PTGS2 (0.76) PTGS2CYP19A1CA1CA2CA9
SCHEMBL19829356 0.83 PTGS2 (0.57) PTGS2CA1CA2CA9GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4920221-A CENTRAL NERVOUS SYSTEM ACTIVE AGENTS PFIZER INC. (US) 1990-04-24 US disclosed
US-4642373-A Substituted dodecahydrotripheylenes, and decahydropyrrolo[1,2-f]phenanthridines as CNS agents PFIZER INC. (US) 1987-02-10 US disclosed
US-4576964-A ANALGESICS, ANTIEMETICS PFIZER INC. (US) 1986-03-18 US disclosed
US-4476131-A ANTIEMETICS, ANALGESICS PFIZER INC. (US) 1984-10-09 US disclosed
US-4473704-A ANALGESICS, ANTIEMETICS PFIZER INC. (US) 1984-09-25 US disclosed