SCHEMBL10474271

SCHEMBL10474271

O=C(O)/C=C/c1cccc2c1O2

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.68
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
NFKB1 P19838 1/20 0.52
CA4 P22748 1/20 0.52
HTT P42858 1/20 0.45
MAPT P10636 1/20 0.45
PARP1 P09874 1/20 0.44
HCAR2 Q8TDS4 2/20 0.44
HDAC3 O15379 1/20 0.44
TNKS O95271 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10474273 1.00 KDM4E (0.68) KDM4ECA1CA2NFKB1CA4
SCHEMBL2855381 0.83 MAPT (0.53) KDM4ENFKB1MAPTLMNAMAOB
SCHEMBL1536573 0.81 KDM4E (1.00) KDM4ECA1CA2NFKB1CA4
SCHEMBL162076 0.81 KDM4E (0.77) KDM4ECA1CA2NFKB1CA4
SCHEMBL1536574 0.81 KDM4E (1.00) KDM4ECA1CA2NFKB1CA4
SCHEMBL162075 0.81 KDM4E (0.77) KDM4ECA1CA2NFKB1CA4
SCHEMBL474092 0.80 ALDH1A1 (0.46) KDM4ECA1CA2MAPTMAOB
SCHEMBL474093 0.80 ALDH1A1 (0.46) KDM4ECA1CA2MAPTMAOB
SCHEMBL7485678 0.78 KDM4E (0.88) KDM4ECA1CA2NFKB1CA4
SCHEMBL8488847 0.77 KDM4E (0.91) KDM4ECA1CA2NFKB1CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4973696-A Stereoselective process for preparing optically active alpha, beta-disubstituted carbonyl compounds ZAMBON S.P.A. (IT) 1990-11-27 US disclosed
EP-0236566-A2 Stereoselective process for preparing optically active alpha, beta-disubstituted carbonyl compounds ZAMBON S.p.A. (IT) 1987-09-16 EP disclosed