SCHEMBL10475641

SCHEMBL10475641

COC(=O)C1=C(C)NC(C)=C(C(=O)O)C1c1cccc(-n2ccnc2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.47
CACNA1B Q00975 2/20 0.47
CACNA1F O60840 4/20 0.47
CACNA1D Q01668 4/20 0.47
CACNA1S Q13698 4/20 0.47
CACNA1C Q13936 4/20 0.47
PDE1C Q14123 2/20 0.47
HTT P42858 1/20 0.46
HIF1A Q16665 3/20 0.45
MEN1 O00255 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
KMT2A Q03164 2/20 0.45
MAPT P10636 2/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
MAPK1 P28482 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10475638 0.96 CACNA1F (0.50) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7268117 0.93 IDO1 (0.47) CACNA1BCYP3A4
SCHEMBL7275109 0.90 ADORA3 (0.59) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL8781999 0.89 IDO1 (0.43) CACNA1BCYP3A4
SCHEMBL8782178 0.87 CACNA1B (0.42) CACNA1B
SCHEMBL30357940 0.85 CACNA1F (0.54) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7269131 0.85 CACNA1F (0.54) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL8928204 0.83 CACNA1C (0.40) CACNA1BCACNA1CPDE1CMAPTLMNA
SCHEMBL10374259 0.80 CYP2C9 (0.42) ADORA3CACNA1BCACNA1CPDE1CHIF1A
SCHEMBL10374261 0.80 CACNA1B (0.43) ADORA3CACNA1BCACNA1FCACNA1DCACNA1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1990006923-A1 IMIDAZOLYL AND PYRIDYL DERIVATIVES OF PHENYL SUBSTITUTED 1,4-DIHYDRO-PYRIDINES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1990-06-28 WO claimed