SCHEMBL8928204

SCHEMBL8928204

CC1=C(C#N)C(c2cccc(-n3ccnc3)c2)C(C(=O)O)=C(C)N1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 3/20 0.40
POLB P06746 2/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PDE2A O00408 1/20 0.40
PDE1A P54750 1/20 0.40
PDE1B Q01064 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE1C Q14123 1/20 0.40
PDE3A Q14432 1/20 0.40
IDO1 P14902 1/20 0.40
GAA P10253 2/20 0.39
ADH5 P11766 1/20 0.39
LMNA P02545 1/20 0.39
GABRA1 P14867 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
ALDH1A1 P00352 4/20 0.38
PKM P14618 1/20 0.38
HSD17B10 Q99714 3/20 0.37
KDM4E B2RXH2 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8860432 0.90 POLB (0.49) POLBMAPK1SMN1; SMN2PDE2APDE1A
SCHEMBL7268117 0.90 IDO1 (0.47) IDO1ADH5CACNA1BPDE4APDE4B
Hydrochloric Acid SCHEMBL8928281 0.88 POLB (0.48) POLBMAPK1SMN1; SMN2PDE2APDE1A
SCHEMBL8928277 0.88 CACNA1C (0.54) CACNA1CALDH1A1MAPT
SCHEMBL8928241 0.87 KDM4E (0.53) CACNA1CGAALMNAALDH1A1HSD17B10
SCHEMBL8781999 0.85 IDO1 (0.43) IDO1ADH5CACNA1BPDE4APDE4B
SCHEMBL10475641 0.83 ADORA3 (0.47) CACNA1CPOLBMAPK1PDE1CLMNA
SCHEMBL8782178 0.78 CACNA1B (0.42) IDO1CACNA1BPDE4APDE4BPDE4C
SCHEMBL10475638 0.78 CACNA1F (0.50) CACNA1CPOLBMAPK1SMN1; SMN2PDE1C
SCHEMBL7273476 0.77 CACNA1F (0.53) CACNA1CPOLBMAPK1SMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP disclosed