SCHEMBL10478166

SCHEMBL10478166

CN1CCC(c2ccccc2)(c2nc(-c3ccccc3)no2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.49
OPRM1 P35372 1/20 0.49
HTT P42858 1/20 0.47
MAPT P10636 2/20 0.44
NOTUM Q6P988 1/20 0.43
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42
NR1H4 Q96RI1 1/20 0.41
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
CHRNA7 P36544 1/20 0.40
CYP2D6 P10635 1/20 0.39
KCNH2 Q12809 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10478397 0.83 OPRM1 (0.51) DRD4OPRM1CHRNA7CYP2D6KCNH2
SCHEMBL10099948 0.83 S1PR1 (0.56) HTTNOTUMS1PR1S1PR3NR1H4
Hydrochloric Acid SCHEMBL10478268 0.82 OPRM1 (0.50) DRD4OPRM1CHRNA7CYP2D6KCNH2
SCHEMBL10620938 0.81 OPRM1 (0.53) OPRM1HTTMAPTNOTUMS1PR1
Hydrochloric Acid SCHEMBL10478033 0.80 OPRM1 (0.51) OPRM1HTTNOTUMS1PR1S1PR3
Oxalic Acid SCHEMBL10478220 0.78 MAPT (0.44) HTTMAPTNPC1RAB9A
Oxalic Acid SCHEMBL10478270 0.78 MAPT (0.39) DRD4OPRM1MAPTS1PR1S1PR3
Hydrochloric Acid SCHEMBL10478080 0.78 OPRM1 (0.46) DRD4OPRM1NR1H4CYP2D6KCNH2
Oxalic Acid SCHEMBL10478394 0.78 KMT2A (0.43) OPRM1HCRTR1HCRTR2
Oxalic Acid SCHEMBL10478168 0.77 LMNA (0.42) DRD4OPRM1MAPTHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4845095-A ANALGESICS, NEUROLEPTICS A/S FERROSAN (DK) 1989-07-04 US claimed
EP-0285032-A1 4-Phenylpiperidine compounds and their preparation and use A/S FERROSAN (DK) 1988-10-05 EP claimed
US-4845095-A ANALGESICS, NEUROLEPTICS A/S FERROSAN (DK) 1989-07-04 US disclosed