SCHEMBL10478397

SCHEMBL10478397

Cc1noc(C2(c3ccccc3)CCN(C)CC2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.51
DRD4 P21917 1/20 0.51
SIGMAR1 Q99720 3/20 0.41
DRD2 P14416 2/20 0.41
KCNH2 Q12809 2/20 0.40
CHRM2 P08172 2/20 0.40
CYP2D6 P10635 2/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
CHRM1 P11229 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
SLC22A1 O15245 1/20 0.38
SLC6A4 P31645 1/20 0.38
ADRA1A P35348 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10478268 0.99 OPRM1 (0.50) OPRM1DRD4SIGMAR1DRD2KCNH2
SCHEMBL10478166 0.83 DRD4 (0.49) OPRM1DRD4SIGMAR1KCNH2CYP2D6
SCHEMBL10478243 0.81 OPRM1 (0.54) OPRM1SIGMAR1DRD2KCNH2SLC6A4
Hydrochloric Acid SCHEMBL10478080 0.80 OPRM1 (0.46) OPRM1DRD4SIGMAR1DRD2KCNH2
Hydrochloric Acid SCHEMBL10477989 0.78 OPRM1 (0.43) OPRM1DRD4SIGMAR1DRD2KCNH2
Oxalic Acid SCHEMBL10478016 0.77 ACKR3 (0.45) DRD2
Oxalic Acid SCHEMBL10478225 0.77 KCNA3 (0.41) OPRM1ADRA1AOPRD1OPRK1
SCHEMBL11738164 0.76 OPRM1 (0.77) OPRM1DRD4SIGMAR1DRD2KCNH2
Hydrochloric Acid SCHEMBL11747049 0.74 OPRM1 (0.74) OPRM1DRD4SIGMAR1DRD2KCNH2
SCHEMBL17001809 0.73 CHRM2 (0.44) CHRM2CHRM1SLC6A4OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4845095-A ANALGESICS, NEUROLEPTICS A/S FERROSAN (DK) 1989-07-04 US disclosed
EP-0285032-A1 4-Phenylpiperidine compounds and their preparation and use A/S FERROSAN (DK) 1988-10-05 EP disclosed