SCHEMBL10484241

SCHEMBL10484241

CCOc1cc2c3ccccc3ccc2c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPRT1 P00492 4/20 0.50
ALOX5 P09917 1/20 0.49
ADORA1 P30542 2/20 0.46
ADORA2A P29274 1/20 0.46
ALDH1A1 P00352 5/20 0.44
HSD17B10 Q99714 2/20 0.43
CYP2A6 P11509 1/20 0.43
TSHR P16473 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
TLR8 Q9NR97 1/20 0.42
HIF1A Q16665 1/20 0.42
CYP1B1 Q16678 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9872788 0.87 HPRT1 (0.52) HPRT1ALOX5ALDH1A1CYP2A6TSHR
SCHEMBL21122175 0.87 HPRT1 (0.52) HPRT1ALOX5ALDH1A1CYP2A6TSHR
SCHEMBL1127908 0.87 TLR8 (0.50) ALOX5ADORA1ADORA2AALDH1A1HSD17B10
SCHEMBL27718961 0.81 HPRT1 (0.48) HPRT1ALOX5ALDH1A1HSD17B10CYP2A6
SCHEMBL755728 0.79 ALOX5 (0.47) HPRT1ALOX5ALDH1A1HSD17B10CYP2A6
SCHEMBL30726470 0.79 ALOX5 (0.47) HPRT1ALOX5ALDH1A1HSD17B10CYP2A6
Chrysene SCHEMBL17075382 0.77 HPRT1 (0.64) HPRT1ALDH1A1HSD17B10CYP2A6TSHR
SCHEMBL12227908 0.76 MAPK1 (0.50) HPRT1ALOX5ALDH1A1HSD17B10TDP1
SCHEMBL30142113 0.76 ALOX5 (0.65) ALOX5ALDH1A1HSD17B10TSHRTDP1
SCHEMBL11882375 0.76 HPRT1 (0.56) HPRT1ALDH1A1HSD17B10CYP2A6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4829090-A SECONDARY AMINES, ANTITUMOR BURROUGHS WELLCOME CO. (US) 1989-05-09 US disclosed
US-4810727-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1989-03-07 US disclosed
US-4719048-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
US-4719046-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
EP-0125702-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1987-08-12 EP disclosed
EP-0125702-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP disclosed