SCHEMBL10484459

SCHEMBL10484459

COC(=O)c1cc(C(=O)OC)cc([P+](C)(c2ccccc2)c2ccccc2)c1.Cc1ccc(S(=O)(=O)[O-])cc1

nearest known ligand 0.45

Known targets — ChEMBL curated mechanism

CHRM1CHRM2CHRM3CHRM4CHRM5SLC6A2dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TCF4 P15884 1/20 0.45
CTNNB1 P35222 1/20 0.45
GAA P10253 2/20 0.44
CYP2C9 P11712 2/20 0.43
TDP1 Q9NUW8 2/20 0.42
TSHR P16473 1/20 0.40
PTGS2 P35354 1/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
KDM4E B2RXH2 2/20 0.38
PPARA Q07869 1/20 0.38
PKM P14618 1/20 0.38
TP53 P04637 2/20 0.38
LMNA P02545 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9634061 0.90 TDP1 (0.51) TCF4CTNNB1GAACYP2C9TDP1
SCHEMBL7733944 0.90 TDP1 (0.51) TCF4CTNNB1GAACYP2C9TDP1
SCHEMBL3137310 0.89 TSHR (0.45) TCF4CTNNB1GAATSHRPTGS2
SCHEMBL10484394 0.85 TSHR (0.45) GAATSHRPTGS2MAPTALDH1A1
SCHEMBL10484503 0.85 TSHR (0.45) GAATSHRPTGS2MAPTALDH1A1
SCHEMBL10484442 0.84 TDP1 (0.57) TCF4CTNNB1GAACYP2C9TDP1
SCHEMBL128521 0.81 CA12 (0.44) GAACYP2C9TDP1MAPTALDH1A1
SCHEMBL9634065 0.80 CA12 (0.41) GAACYP2C9TSHRPTGS2ALDH1A1
Tetraphenylphosphonium SCHEMBL6735186 0.79 TSHR (0.46) TCF4CTNNB1GAATSHRPTGS2
SCHEMBL10484434 0.78 TDP1 (0.49) TCF4CTNNB1GAACYP2C9TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4496643-A PHOSPHONIUM, ARSONIUM, OR STIBONIUM COMPOUND IN BINDER AS TONER AND FLUOROCARBON CARRIER COATED PARTICLES EASTMAN KODAK COMPANY (US) 1985-01-29 US claimed
US-4855396-A BINDER/CHARGE AGENT IN ELECTROSTATOGRAPHIC TONER PARTICLES EASTMAN KODAK COMPANY (US) 1989-08-08 US disclosed
US-4837394-A CHARGE CONTROL AGENTS EASTMAN KODAK COMPANY (US) 1989-06-06 US disclosed
EP-0161128-A1 Two-component dry electrostatic developer composition EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1985-11-13 EP disclosed