SCHEMBL10487407

SCHEMBL10487407

CCOC(=O)[C@@H](C)Oc1ccc(F)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.51
EPHX2 P34913 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
LMNA P02545 1/20 0.50
PPOX P50336 1/20 0.46
ALDH2 P05091 1/20 0.45
GAA P10253 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TSHR P16473 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 2/20 0.42
NPC1 O15118 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10714951 1.00 KMT2A (0.51) KMT2AEPHX2L3MBTL1LMNAPPOX
SCHEMBL25577860 0.86 L3MBTL1 (0.54) KMT2AEPHX2L3MBTL1LMNAPPOX
SCHEMBL5208842 0.86 L3MBTL1 (0.54) KMT2AEPHX2L3MBTL1LMNAPPOX
SCHEMBL10487443 0.86 KMT2A (0.55) KMT2AEPHX2L3MBTL1LMNAALDH2
SCHEMBL25577858 0.86 L3MBTL1 (0.54) KMT2AEPHX2L3MBTL1LMNAPPOX
SCHEMBL13744595 0.85 KMT2A (0.53) KMT2AEPHX2L3MBTL1LMNAALDH2
SCHEMBL15261678 0.83 TSHR (0.43) KMT2AL3MBTL1TSHRKDM4EMAPT
SCHEMBL10022852 0.83 EPHX2 (0.66) KMT2AEPHX2L3MBTL1LMNAGAA
SCHEMBL5204883 0.83 EPHX2 (0.66) KMT2AEPHX2L3MBTL1LMNAGAA
SCHEMBL17710797 0.81 TDP1 (0.56) EPHX2GAATDP1TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1015545-B preparation method of glycolic acid derivative for treating diabetic complications PFIZER (US) 1992-02-19 CN disclosed
US-4853410-A Hydroxyacetic acid derivatives for the treatment of diabetic complications PFIZER INC. (US) 1989-08-01 US disclosed
CN-87100191-A The hydroxy acid derivative of treatment diabetic complication 1987-09-09 CN disclosed
WO-1987004344-A1 HYDROXYACETIC ACID DERIVATIVES FOR THE TREATMENT OF DIABETIC COMPLICATIONS PFIZER INC. (US) 1987-07-30 WO disclosed
EP-0230379-A2 Chroman- and thiochroman-4-acetic acids useful in the treatment of diabetic complications PFIZER INC. (US) 1987-07-29 EP disclosed