SCHEMBL10488176

SCHEMBL10488176

CCCc1cc(CCCCOCCCCCNCC(O)c2ccc(O)c(NS(C)(=O)=O)c2)ccc1C(=O)O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 16/20 0.63
CHRM3 P20309 1/20 0.63
ADRB3 P13945 18/20 0.58
ADRB1 P08588 15/20 0.58
KDM4E B2RXH2 1/20 0.54
MEN1 O00255 1/20 0.54
GMNN O75496 1/20 0.54
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
TP53 P04637 1/20 0.54
CYP3A4 P08684 1/20 0.54
HPGD P15428 1/20 0.54
NFKB1 P19838 1/20 0.54
MAPK1 P28482 1/20 0.54
THPO P40225 1/20 0.54
MTOR P42345 1/20 0.54
RAB9A P51151 1/20 0.54
BLM P54132 1/20 0.54
PMP22 Q01453 1/20 0.54
KMT2A Q03164 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10706286 0.87 ADRB2 (0.66) ADRB2CHRM3ADRB3ADRB1KDM4E
SCHEMBL10488179 0.84 ADRB2 (0.60) ADRB2CHRM3ADRB3ADRB1KDM4E
SCHEMBL10488131 0.83 ADRB3 (0.71) ADRB2CHRM3ADRB3ADRB1
SCHEMBL10488196 0.83 ADRB2 (0.65) ADRB2CHRM3ADRB3ADRB1KDM4E
SCHEMBL10488095 0.83 ADRB2 (0.65) ADRB2CHRM3ADRB3ADRB1KDM4E
SCHEMBL10488200 0.82 ADRB2 (0.62) ADRB2CHRM3ADRB3ADRB1KDM4E
SCHEMBL10488093 0.82 ADRB2 (0.58) ADRB2CHRM3ADRB3ADRB1KDM4E
SCHEMBL10488552 0.82 ADRB2 (0.64) ADRB2CHRM3ADRB3ADRB1KDM4E
SCHEMBL10488154 0.81 ADRB2 (0.61) ADRB2CHRM3ADRB3ADRB1
Acetic Acid SCHEMBL10488094 0.81 ADRB2 (0.61) ADRB2CHRM3ADRB3ADRB1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0178919-B1 AMINOPHENOL DERIVATIVES GLAXO GROUP LIMITED (GB) 1988-12-21 EP claimed
US-4853382-A TREATING ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1989-08-01 US disclosed
EP-0178919-B1 AMINOPHENOL DERIVATIVES GLAXO GROUP LIMITED (GB) 1988-12-21 EP disclosed
US-4730008-A STIMULANT FOR BETA-ADRENORECEPTORS GLAXO GROUP LIMITED (GB) 1988-03-08 US disclosed