SCHEMBL10488702

SCHEMBL10488702

CSc1ccccc1NC(=S)NN

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.59
MAPT P10636 2/20 0.58
LMNA P02545 2/20 0.58
KDM4E B2RXH2 1/20 0.58
GAA P10253 1/20 0.57
HTT P42858 1/20 0.56
KMT2A Q03164 1/20 0.52
IDO1 P14902 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5526225 0.81 L3MBTL1 (0.55) ALDH1A1MAPTLMNAKDM4EGAA
SCHEMBL5434789 0.77 MAPT (0.61) ALDH1A1MAPTLMNAKDM4EGAA
SCHEMBL29488187 0.77 MAPT (0.61) ALDH1A1MAPTLMNAKDM4EGAA
SCHEMBL4210466 0.75 KMT2A (0.62) ALDH1A1MAPTLMNAHTTKMT2A
SCHEMBL7349 0.73 ALDH1A1 (0.47) ALDH1A1MAPTLMNAKMT2A
SCHEMBL29573636 0.73 ALDH1A1 (0.47) ALDH1A1MAPTLMNAKMT2A
SCHEMBL23220327 0.73 ALDH1A1 (0.61) ALDH1A1MAPTLMNAKDM4EGAA
SCHEMBL5430219 0.73 ALDH1A1 (1.00) ALDH1A1MAPTLMNAKDM4EGAA
SCHEMBL29488194 0.73 ALDH1A1 (1.00) ALDH1A1MAPTLMNAKDM4EGAA
SCHEMBL15165726 0.73 MAPT (0.56) ALDH1A1MAPTLMNAKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4871737-A 3-Amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants muscle relaxants and anxiolytics A. H. ROBINS COMPANY, INCORPORATED (US) 1989-10-03 US disclosed
EP-0315433-A2 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics A.H. ROBINS COMPANY, INCORPORATED (US) 1989-05-10 EP disclosed
US-4826866-A 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics A. H. ROBINS COMPANY, INCORPORATED (US) 1989-05-02 US disclosed