SCHEMBL10498917

SCHEMBL10498917

Cc1cc(C)nc(N(C(N)=NN(C)C)S(=O)(=O)c2ccccc2Cl)n1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.54
SMN1; SMN2 Q16637 1/20 0.51
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
GAA P10253 2/20 0.39
LMNA P02545 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PGR P06401 1/20 0.35
MAPT P10636 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTT P42858 1/20 0.34
HCRTR2 O43614 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10867034 0.91 SMN1; SMN2 (0.67) KDM4ESMN1; SMN2CYP1A2CYP3A4CYP2D6
SCHEMBL9591445 0.90 KDM4E (0.58) KDM4ESMN1; SMN2CYP1A2CYP3A4CYP2D6
SCHEMBL10865751 0.88 KDM4E (0.39) KDM4ESMN1; SMN2MEN1KMT2AMAPT
SCHEMBL10867587 0.85 SMN1; SMN2 (0.56) KDM4ESMN1; SMN2CYP1A2CYP3A4CYP2D6
SCHEMBL10568364 0.83 MEN1 (0.51) KDM4ESMN1; SMN2CYP1A2CYP3A4CYP2D6
SCHEMBL9478178 0.82 KDM4E (0.50) KDM4ESMN1; SMN2CYP1A2CYP3A4CYP2D6
SCHEMBL10502876 0.81 CA1 (0.44) KDM4ESMN1; SMN2MEN1KMT2AMAPT
SCHEMBL9735397 0.81 SMN1; SMN2 (0.69) KDM4ESMN1; SMN2CYP1A2CYP3A4CYP2D6
SCHEMBL10688914 0.81 HCRTR1 (0.43) KDM4ESMN1; SMN2HCRTR2
SCHEMBL10865204 0.78 ALDH1A1 (0.41) KDM4ESMN1; SMN2CYP3A4LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4880932-A PLANT GROWTH REGULATORS, HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1989-11-14 US disclosed
EP-0121082-B1 GUANIDIN DERIVATIVES BAYER AG (DE) 1989-11-08 EP disclosed
US-4844730-A PLANT GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1989-07-04 US disclosed
US-4797484-A REACTING GUANIDINE DERIVATIVE WITH SULPHONYL HALIDE BAYER AKTIENGESELLSCHAFT (DE) 1989-01-10 US disclosed
US-4743294-A N'-(substituted-1,3,5-triazin-2-yl)-N\"-amino-N\"'-(substituted-benzenesulphonyl)-guanidines as herbicides BAYER AKTIENGESELLSCHAFT (DE) 1988-05-10 US disclosed
US-4725305-A PLANT GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1988-02-16 US disclosed
US-4725303-A N'-(substituted-pyrimidin-2-yl)-N\"-amino-N\"'-(substituted-benzenesulphonyl)-guanidines as herbicides BAYER AKTIENGESELLSCHAFT (DE) 1988-02-16 US disclosed
US-4721785-A FOR THE 2-GUANIDINE DERIVATIVE HERBICIDE PRODUCTS BAYER AKTIENGESELLSCHAFT (DE) 1988-01-26 US disclosed
US-4602938-A N'-(substituted-pyrimidin-2-yl)-N\"-substituted-N\",N\"'-bis-(substituted-benzenesulphonyl)-guanidines as herbicides BAYER AKTIENGESELLSCHAFT (DE) 1986-07-29 US disclosed
EP-0121082-A1 Guanidin derivatives BAYER AG (DE) 1984-10-10 EP disclosed