SCHEMBL10503157

SCHEMBL10503157

COc1nc(C)nc(NC(NS(=O)(=O)c2ccccc2SC)=[N+](OC)S(=O)(=O)c2ccccc2SC)n1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.30
GAA P10253 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10867785 0.86 NPC1 (0.36) ALDH1A1KDM4ENPC1MAPT
SCHEMBL10563335 0.85 KDM4E (0.43) ALDH1A1KDM4ENPC1MAPTGAA
SCHEMBL9684325 0.79 MAPT (0.46) ALDH1A1KDM4ENPC1MAPT
SCHEMBL9480849 0.78 POLB (0.34) ALDH1A1KDM4ENPC1MAPT
SCHEMBL10918288 0.77 SLC22A12 (0.39)
SCHEMBL10500864 0.76 SLC22A12 (0.43) ALDH1A1
SCHEMBL10868380 0.76 ALDH1A1 (0.37) ALDH1A1MAPT
SCHEMBL10761883 0.72 HPGD (0.45) ALDH1A1NPC1MAPTGAAHTT
SCHEMBL11170537 0.72 MAPT (0.43) ALDH1A1KDM4ENPC1MAPTGAA
SCHEMBL10756516 0.72 FBP1 (0.39) ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4797484-A REACTING GUANIDINE DERIVATIVE WITH SULPHONYL HALIDE BAYER AKTIENGESELLSCHAFT (DE) 1989-01-10 US disclosed