SCHEMBL10508908

SCHEMBL10508908

O=C(O)/C(=C\NC1CC1)C(=O)c1c(F)c(F)c(F)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
TAS1R3 Q7RTX0 4/20 0.32
TAS1R1 Q7RTX1 3/20 0.32
TAS1R2 Q8TE23 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10508912 1.00 CES2 (0.32) CES2CES1TAS1R3TAS1R1TAS1R2
SCHEMBL9377242 0.86
SCHEMBL9377247 0.86
SCHEMBL10774464 0.82 ALDH1A1 (0.41)
SCHEMBL9689331 0.79 CRBN (0.37) CES2CES1
SCHEMBL9689334 0.79 CRBN (0.37) CES2CES1
SCHEMBL7510222 0.79 POLB (0.40) TAS1R3TAS1R1TAS1R2
SCHEMBL7510218 0.79 POLB (0.40) TAS1R3TAS1R1TAS1R2
SCHEMBL1345391 0.78 CYP2D6 (0.38) TAS1R3TAS1R1TAS1R2
SCHEMBL9562436 0.78 CYP2D6 (0.38) TAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0202763-B1 5,6-DIFLUORONAPHTHYRIDINES AND 5,6,8-TRIFLUORO-QUINOLINES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1989-11-08 EP disclosed
US-4657913-A Trifluoro- quinoline -3- carboxylic acids and their use as anti-bacterial agents WARNER-LAMBERT COMPANY (US) 1987-04-14 US disclosed
EP-0202763-A1 5,6-Difluoronaphthyridines and 5,6,8-trifluoro-quinolines as antibacterial agents WARNER-LAMBERT COMPANY (US) 1986-11-26 EP disclosed