SCHEMBL10509367

SCHEMBL10509367

NC(F)Cc1ccc(O)cc1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.61
SLC6A2 P23975 2/20 0.61
SLC7A5 Q01650 1/20 0.55
ESR1 P03372 6/20 0.48
ESR2 Q92731 6/20 0.48
ABAT P80404 1/20 0.48
OPRK1 P41145 1/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTR3A P46098 1/20 0.44
BACE1 P56817 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19692716 0.81 PRSS1 (0.41) TAAR1SLC6A2SLC7A5
SCHEMBL8014472 0.80 TAAR1 (0.67) TAAR1SLC6A2SLC7A5ESR1ESR2
SCHEMBL15951398 0.80 TAAR1 (0.67) TAAR1SLC6A2SLC7A5ESR1ESR2
SCHEMBL5570367 0.80 TAAR1 (0.54) TAAR1SLC6A2SLC7A5ESR1ESR2
SCHEMBL5332232 0.79 TAAR1 (0.59) TAAR1SLC6A2SLC7A5ESR1ESR2
SCHEMBL21357615 0.78 TAAR1 (0.64) TAAR1SLC6A2SLC7A5ESR1ESR2
SCHEMBL14797209 0.78 LOXL2 (0.50) TAAR1
SCHEMBL21632218 0.78 TAAR1 (0.64) TAAR1SLC6A2SLC7A5ESR1ESR2
SCHEMBL1048764 0.78 TAAR1 (0.64) TAAR1SLC6A2SLC7A5ESR1ESR2
SCHEMBL22074724 0.77 TAAR1 (0.57) TAAR1SLC6A2SLC7A5ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0163948-B1 PROCESS FOR PRODUCING AN INDOLINE IHARA CHEMICAL IND CO 1989-08-16 EP disclosed
US-4673749-A CYCLIZATION OF 2-HOLOGENO PHENETHYLAMINES WITH COPPER CATALYS T AND ALKALI DEHYROHALOGENATING AGENT IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 1987-06-16 US disclosed
EP-0163948-A1 Process for producing an indoline IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 1985-12-11 EP disclosed
US-4280958-A COPPER-TYPE CATALYST USED IN CYCLIZATION OF A HALOGENOPHENETHYLAMINE IN THE PRESENCE OF AN AMINE IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 1981-07-28 US disclosed
US-4159271-A CYCLIZATION OF A 2-HALOGENOPHENETHYLAMINE IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 1979-06-26 US disclosed