SCHEMBL10510260

SCHEMBL10510260

Nc1cccc(Cc2c(F)cccc2F)c1N

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.42
TAAR1 Q96RJ0 3/20 0.38
HTT P42858 2/20 0.36
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CD44 P16070 1/20 0.35
IDO1 P14902 2/20 0.35
AR P10275 1/20 0.33
LMNA P02545 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3132841 0.80 CD44 (0.46) ALDH1A1L3MBTL1CD44
SCHEMBL11780183 0.80 TAAR1 (0.47) MPOTAAR1HTTALDH1A1NPC1
SCHEMBL1750348 0.77 TAAR1 (0.43) MPOTAAR1ALDH1A1L3MBTL1IDO1
SCHEMBL31470103 0.74 HTT (0.51) TAAR1HTTNPC1L3MBTL1IDO1
SCHEMBL2356316 0.74 CYP3A4 (0.41) ALDH1A1L3MBTL1CD44AR
SCHEMBL11778004 0.73 ALDH1A1 (0.47) MPOTAAR1HTTALDH1A1NPC1
SCHEMBL601969 0.73
SCHEMBL29803091 0.73
SCHEMBL5205493 0.72 TAAR1 (0.46) MPOTAAR1HTTALDH1A1NPC1
SCHEMBL28047780 0.72 TAAR1 (0.47) MPOTAAR1NPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0145037-B1 N-(BICYCLIC HETEROCYCLYL)-4-PIPERIDINAMINES JANSSEN PHARMACEUTICA N.V. (BE) 1989-01-18 EP disclosed
EP-0145037-A2 N-(bicyclic heterocyclyl)-4-piperidinamines JANSSEN PHARMACEUTICA N.V. (BE) 1985-06-19 EP disclosed