SCHEMBL10521561

SCHEMBL10521561

CC(C)CCC(=O)CNC(=O)OC(C)(C)CBr

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
CA1 P00915 2/20 0.32
KCNA5 P22460 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24928346 0.84 MEN1 (0.46) MEN1GAAKMT2ACA1KCNA5
SCHEMBL7265384 0.74 HPGD (0.38) MEN1KMT2A
SCHEMBL21582671 0.70 MEN1 (0.39) MEN1GAAKMT2ACA1KCNA5
SCHEMBL23354478 0.69 CYP2D6 (0.48) CA1
SCHEMBL31466178 0.68 CYP2D6 (0.39) MEN1GAAKMT2ACA1
SCHEMBL16153117 0.68 RIPK1 (0.39) CA1
SCHEMBL13306481 0.66 TDP1 (0.46) MEN1GAAKMT2ACA1
SCHEMBL19750462 0.66 RECQL (0.44) MEN1GAAKMT2ACA1
SCHEMBL3686909 0.65 TDP1 (0.44) MEN1GAAKMT2ACA1
SCHEMBL8535486 0.65 TDP1 (0.53) MEN1GAAKMT2ACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4829053-A Amino acid derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1989-05-09 US disclosed
EP-0262318-A2 Renin-inhibiting amino acid derivatives MERCK PATENT GmbH (DE) 1988-04-06 EP disclosed